# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3979322 | 13 | IC50 | = | 0.18 | nM | ALA3855037 | 9.74 | nM | Homo sapiens | ||
2. | ALA3979322 | 13 | IC50 | = | 9.2 | nM | ALA3855038 | 8.04 | nM | Rattus norvegicus | ||
3. | ALA3979322 | 13 | Drug uptake | = | 60 | nM | ALA3855051 | nM | ||||
4. | ALA3979322 | 13 | Occ | = | 9 | % | ALA3855049 | % | Rattus norvegicus | |||
5. | ALA3979322 | 13 | Drug uptake | = | 687 | nM | ALA3855048 | nM | ||||
6. | ALA3979322 | 13 | Drug uptake | = | 188 | nM | ALA3855047 | nM | ||||
7. | ALA3979322 | 13 | Occ | = | 70 | % | ALA3855045 | % | Rattus norvegicus | |||
8. | ALA3979322 | 13 | Occ | = | 54 | % | ALA3855044 | % | Rattus norvegicus | |||
9. | ALA3979322 | 13 | solubility | = | 0.77 | mg/ml | ALA3855042 | ug.mL-1 | ||||
10. | ALA3979322 | 13 | IC50 | = | 4 | uM | ALA3855039 | 5.40 | nM | Homo sapiens | ||
11. | ALA3979322 | 13 | permeability | = | 4.8 | % | ALA3855036 | % |