| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3980860 | BDBM194644 | IC50 | = | 2 | nM | ALA4835256 | 8.70 | nM | Homo sapiens | ||
| 2. | ALA3980860 | BDBM194644 | IC50 | = | 2 | nM | ALA4835255 | 8.70 | nM | Homo sapiens | ||
| 3. | ALA3980860 | BDBM194644 | Ratio | >= | 10 | ALA4013286 | ||||||
| 4. | ALA3980860 | BDBM194644 | Drug metabolism | 0 | ALA4013285 | Metabolite_Notdetected | Rattus norvegicus | |||||
| 5. | ALA3980860 | BDBM194644 | Activity | = | 53 | % | ALA4013284 | % | Rattus norvegicus | |||
| 6. | ALA3980860 | BDBM194644 | Activity | = | 52 | % | ALA4013283 | % | Rattus norvegicus | |||
| 7. | ALA3980860 | BDBM194644 | Activity | = | 41 | % | ALA4013282 | % | Rattus norvegicus | |||
| 8. | ALA3980860 | BDBM194644 | F | = | 100 | % | ALA4013281 | % | Rattus norvegicus | |||
| 9. | ALA3980860 | BDBM194644 | Vd | = | 4.3 | L/Kg | ALA4013280 | L.kg-1 | Rattus norvegicus | |||
| 10. | ALA3980860 | BDBM194644 | CL | = | 33 | ml/min.kg | ALA4013279 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 11. | ALA3980860 | BDBM194644 | t1/2 | = | 2.6 | hr | ALA4013278 | hr | Rattus norvegicus | |||
| 12. | ALA3980860 | BDBM194644 | t1/2 | = | 1.5 | hr | ALA4013277 | hr | Rattus norvegicus | |||
| 13. | ALA3980860 | BDBM194644 | AUC | = | 22000 | nM.hr | ALA4013276 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 14. | ALA3980860 | BDBM194644 | AUC | = | 1300 | nM.hr | ALA4013275 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 15. | ALA3980860 | BDBM194644 | Cp | < | 5 | nM | ALA4013274 | nM | Rattus norvegicus | |||
| 16. | ALA3980860 | BDBM194644 | Cp | = | 29 | nM | ALA4013273 | nM | Rattus norvegicus | |||
| 17. | ALA3980860 | BDBM194644 | Tmax | = | 0.5 | hr | ALA4013272 | hr | Rattus norvegicus | |||
| 18. | ALA3980860 | BDBM194644 | Cmax | = | 6600 | nM | ALA4013263 | nM | Rattus norvegicus | |||
| 19. | ALA3980860 | BDBM194644 | Cmax | = | 1600 | nM | ALA4013262 | nM | Rattus norvegicus | |||
| 20. | ALA3980860 | BDBM194644 | IC50 | = | 50000 | nM | ALA4013271 | 4.30 | nM | Homo sapiens |
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