# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4059621 | 24 | CI | = | 1.246 | ALA4041626 | ||||||
2. | ALA4059621 | 24 | CI | = | 1.163 | ALA4041625 | ||||||
3. | ALA4059621 | 24 | CI | = | 1.061 | ALA4041624 | ||||||
4. | ALA4059621 | 24 | Activity | = | 28 | ALA4041621 | Salmonella enterica subsp. enterica serovar Typhimurium | |||||
5. | ALA4059621 | 24 | F | = | 0.74 | % | ALA4041618 | % | Rattus norvegicus | |||
6. | ALA4059621 | 24 | t1/2 | = | 2.25 | hr | ALA4041617 | hr | Rattus norvegicus | |||
7. | ALA4059621 | 24 | t1/2 | = | 0.92 | ug ml-1 | ALA4041620 | ug ml-1 | Rattus norvegicus | |||
8. | ALA4059621 | 24 | Cmax | = | 1.68 | ug ml-1 | ALA4041619 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
9. | ALA4059621 | 24 | Cmax | = | 0.017 | ug ml-1 | ALA4041616 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
10. | ALA4059621 | 24 | Stability | = | 87.2 | % | ALA4041615 | % | Rattus norvegicus | |||
11. | ALA4059621 | 24 | EC50 | = | 0.032 | nM | ALA4041600 | 10.49 | nM | |||
12. | ALA4059621 | 24 | EC50 | = | 0.882 | nM | ALA4041601 | 9.05 | nM | |||
13. | ALA4059621 | 24 | Activity | > | 30 | uM | ALA4041602 | uM | Homo sapiens | |||
14. | ALA4059621 | 24 | INH | = | 18.7 | % | ALA4041603 | % | Homo sapiens | |||
15. | ALA4059621 | 24 | Stability | = | 92.6 | % | ALA4041604 | % | Homo sapiens | |||
16. | ALA4059621 | 24 | Activity | = | 29 | ALA4041605 | Salmonella enterica subsp. enterica serovar Typhimurium | |||||
17. | ALA4059621 | 24 | Activity | = | 110 | ALA4041611 | Salmonella enterica subsp. enterica serovar Typhimurium | |||||
18. | ALA4059621 | 24 | Activity | = | 125 | ALA4041612 | Salmonella enterica subsp. enterica serovar Typhimurium | |||||
19. | ALA4059621 | 24 | CI | = | 0.98 | ALA4041614 |