# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4060185 | 8k | Efficacy | = | 1063 | % | ALA4367978 | % | Rattus norvegicus | |||
2. | ALA4060185 | 8k | FC | = | 20 | ALA4219590 | Homo sapiens | |||||
3. | ALA4060185 | 8k | FC | = | 2 | ALA4219589 | Homo sapiens | |||||
4. | ALA4060185 | 8k | FC | = | 2 | ALA4219588 | Homo sapiens | |||||
5. | ALA4060185 | 8k | FC | = | 5 | ALA4219587 | Homo sapiens | |||||
6. | ALA4060185 | 8k | FC | = | 8 | ALA4219586 | Homo sapiens | |||||
7. | ALA4060185 | 8k | FC | = | 10 | ALA4219580 | Homo sapiens | |||||
8. | ALA4060185 | 8k | Ki | = | 1.9 | nM | ALA4219585 | 8.72 | nM | Homo sapiens | ||
9. | ALA4060185 | 8k | Ki | = | 0.3 | nM | ALA4219584 | 9.52 | nM | Homo sapiens | ||
10. | ALA4060185 | 8k | Ki | > | 10 | uM | ALA4219583 | nM | Homo sapiens | |||
11. | ALA4060185 | 8k | Ki | = | 0.2 | nM | ALA4219582 | 9.70 | nM | Homo sapiens | ||
12. | ALA4060185 | 8k | Ki | > | 10 | uM | ALA4219581 | nM | Homo sapiens | |||
13. | ALA4060185 | 8k | Ki | = | 0.2 | nM | ALA4219578 | 9.70 | nM | Homo sapiens | ||
14. | ALA4060185 | 8k | solubility | = | 8.5 | uM | ALA4037811 | nM | ||||
15. | ALA4060185 | 8k | solubility | = | 6.4 | uM | ALA4037810 | nM | ||||
16. | ALA4060185 | 8k | Stability | = | 69.2 | % | ALA4037809 | % | Mus musculus | |||
17. | ALA4060185 | 8k | t1/2 | = | 1.9 | hr | ALA4037808 | hr | Mus musculus | |||
18. | ALA4060185 | 8k | Stability | = | 72.5 | % | ALA4037807 | % | Homo sapiens | |||
19. | ALA4060185 | 8k | t1/2 | = | 2.3 | hr | ALA4037806 | hr | Homo sapiens | |||
20. | ALA4060185 | 8k | Activity | 0 | ALA4037852 | Non-Toxic | Mus musculus |