# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4060827 | 41, epimeric mixture | Ki | = | 0.29 | nM | ALA4735354 | 9.54 | nM | Homo sapiens | ||
2. | ALA4060827 | 41, epimeric mixture | Kd(app) | = | 2.1 | uM | ALA4020043 | 5.68 | nM | Homo sapiens | ||
3. | ALA4060827 | 41, epimeric mixture | Kd | = | 0.004 | uM | ALA4020042 | 8.40 | nM | Homo sapiens | ||
4. | ALA4060827 | 41, epimeric mixture | K | = | 0.005 | /s | ALA4020041 | /s | Homo sapiens | |||
5. | ALA4060827 | 41, epimeric mixture | Ki | = | 0.001 | uM | ALA4020039 | 9.15 | nM | Homo sapiens | ||
6. | ALA4060827 | 41, epimeric mixture | K | = | 1.3 | 10'6/M/s | ALA4020040 | 10'6/M/s | Homo sapiens | |||
7. | ALA4060827 | 41, epimeric mixture | CL free | = | 220 | L/hr/kg | ALA4007112 | mL.min-1.kg-1 | Mus musculus | |||
8. | ALA4060827 | 41, epimeric mixture | IC50 | = | 33 | nM | ALA4007111 | 7.48 | nM | Homo sapiens | ||
9. | ALA4060827 | 41, epimeric mixture | IC50 | = | 50 | nM | ALA4007110 | 7.30 | nM | Homo sapiens | ||
10. | ALA4060827 | 41, epimeric mixture | IC50 | = | 33 | nM | ALA4007109 | 7.48 | nM | Homo sapiens | ||
11. | ALA4060827 | 41, epimeric mixture | Ki | = | 0.29 | nM | ALA4007108 | 9.54 | nM | Homo sapiens |