| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4062567 | 1; LJN452 | Activity | = | 98.23 | % | ALA5157313 | % | Homo sapiens | |||
| 2. | ALA4062567 | 1; LJN452 | EC50 | = | 2.64 | nM | ALA5157312 | 8.58 | nM | Homo sapiens | ||
| 3. | ALA4062567 | 1; LJN452 | Activity | = | 118.8 | % | ALA5157311 | % | Homo sapiens | |||
| 4. | ALA4062567 | 1; LJN452 | EC50 | = | 1.1 | nM | ALA5157310 | 8.96 | nM | Homo sapiens | ||
| 5. | ALA4062567 | 1; LJN452 | Activity | 0 | ALA4032786 | Dose-dependent effect | Rattus norvegicus | |||||
| 6. | ALA4062567 | 1; LJN452 | FC | = | 3 | ALA4032677 | Rattus norvegicus | |||||
| 7. | ALA4062567 | 1; LJN452 | FC | = | 15 | ALA4032676 | Rattus norvegicus | |||||
| 8. | ALA4062567 | 1; LJN452 | Activity | 0 | ALA4032675 | Dose-dependent effect | Rattus norvegicus | |||||
| 9. | ALA4062567 | 1; LJN452 | Activity | 0 | ALA4032674 | Dose-dependent effect | Rattus norvegicus | |||||
| 10. | ALA4062567 | 1; LJN452 | Drug metabolism | 0 | ALA4032816 | Metabolite_Notdetected | Canis lupus familiaris | |||||
| 11. | ALA4062567 | 1; LJN452 | Drug metabolism | 0 | ALA4032815 | Metabolite_Notdetected | Rattus norvegicus | |||||
| 12. | ALA4062567 | 1; LJN452 | Drug metabolism | 0 | ALA4032814 | Metabolite_Notdetected | Mus musculus | |||||
| 13. | ALA4062567 | 1; LJN452 | Drug metabolism | 0 | ALA4032813 | Metabolite_Notdetected | Canis lupus familiaris | |||||
| 14. | ALA4062567 | 1; LJN452 | Drug metabolism | 0 | ALA4032812 | Metabolite_Notdetected | Rattus norvegicus | |||||
| 15. | ALA4062567 | 1; LJN452 | Drug metabolism | 0 | ALA4032811 | Metabolite_Notdetected | Mus musculus | |||||
| 16. | ALA4062567 | 1; LJN452 | F | = | 10 | % | ALA4032810 | % | Rattus norvegicus | |||
| 17. | ALA4062567 | 1; LJN452 | Cmax | = | 53 | nM | ALA4032809 | nM | Rattus norvegicus | |||
| 18. | ALA4062567 | 1; LJN452 | AUC | = | 307 | hr.nM | ALA4032808 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 19. | ALA4062567 | 1; LJN452 | Ratio | = | 6 | ALA4032807 | ||||||
| 20. | ALA4062567 | 1; LJN452 | Ratio | = | 14 | ALA4032806 |
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