| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4062760 | 8 | EC50 | = | 5 | nM | ALA5247740 | 8.30 | nM | Homo sapiens | ||
| 2. | ALA4062760 | 8 | F | = | 37 | % | ALA4032673 | % | Rattus norvegicus | |||
| 3. | ALA4062760 | 8 | Cmax | = | 382 | nM | ALA4032672 | nM | Rattus norvegicus | |||
| 4. | ALA4062760 | 8 | AUC | = | 4571 | hr.nM | ALA4032671 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 5. | ALA4062760 | 8 | beta t1/2 | = | 1 | hr | ALA4032670 | hr | Rattus norvegicus | |||
| 6. | ALA4062760 | 8 | Vdss | = | 1.2 | L/Kg | ALA4032669 | L.kg-1 | Rattus norvegicus | |||
| 7. | ALA4062760 | 8 | CL | = | 24 | ml/min.kg | ALA4032668 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 8. | ALA4062760 | 8 | ERH | < | 0.21 | ALA4032667 | Homo sapiens | |||||
| 9. | ALA4062760 | 8 | ERH | < | 0.18 | ALA4032666 | Rattus norvegicus | |||||
| 10. | ALA4062760 | 8 | solubility | = | 70 | uM | ALA4032664 | nM | ||||
| 11. | ALA4062760 | 8 | Efficacy | = | 100 | % | ALA4032663 | % | Homo sapiens | |||
| 12. | ALA4062760 | 8 | EC50 | = | 19 | nM | ALA4032662 | 7.72 | nM | Homo sapiens | ||
| 13. | ALA4062760 | 8 | Efficacy | = | 97 | % | ALA4032661 | % | Homo sapiens | |||
| 14. | ALA4062760 | 8 | EC50 | = | 19 | nM | ALA4032660 | 7.72 | nM | Homo sapiens |
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