# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4063082 | 24b | Activity | = | 17 | % | ALA3999943 | % | Rattus norvegicus | |||
2. | ALA4063082 | 24b | AUC | = | 19.65 | ug.hr/ml | ALA3999942 | ng.hr.mL-1 | Rattus norvegicus | |||
3. | ALA4063082 | 24b | Cmax | = | 3.35 | ug ml-1 | ALA3999941 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
4. | ALA4063082 | 24b | Stability | = | 81 | % | ALA3999940 | % | Rattus norvegicus | |||
5. | ALA4063082 | 24b | IC50 | = | 0.002 | uM | ALA3999937 | 8.70 | nM | Homo sapiens | ||
6. | ALA4063082 | 24b | Drug metabolism | 0 | ALA3999936 | Metabolite_Notdetected | Homo sapiens | |||||
7. | ALA4063082 | 24b | logD | = | 4.3 | ALA4044737 | ||||||
8. | ALA4063082 | 24b | IC50 | = | 0.11 | uM | ALA4044731 | 6.96 | nM | Rattus norvegicus | ||
9. | ALA4063082 | 24b | IC50 | = | 0.002 | uM | ALA4044730 | 8.70 | nM | Homo sapiens | ||
10. | ALA4063082 | 24b | solubility | = | 1.8 | ug ml-1 | ALA4044738 | ug.mL-1 | ||||
11. | ALA4063082 | 24b | solubility | = | 1.5 | ug ml-1 | ALA4044739 | ug.mL-1 | ||||
12. | ALA4063082 | 24b | solubility | = | 12 | ug ml-1 | ALA4044740 | ug.mL-1 |