# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4064397 | 16 | FC | = | 7 | ALA4028357 | Mus musculus | |||||
2. | ALA4064397 | 16 | Activity | 0 | ALA4028397 | Non-Toxic | Rattus norvegicus | |||||
3. | ALA4064397 | 16 | Activity | 0 | ALA4028360 | Active | Mus musculus | |||||
4. | ALA4064397 | 16 | IC50 | = | 34.2 | nM | ALA4028335 | 7.47 | nM | Homo sapiens | ||
5. | ALA4064397 | 16 | MTD | = | 75 | mg kg-1 | ALA4028336 | mg kg-1 | Mus musculus | |||
6. | ALA4064397 | 16 | Efficacy | = | -1.2 | % | ALA4028337 | % | Homo sapiens | |||
7. | ALA4064397 | 16 | Efficacy | = | 0.5 | % | ALA4028338 | % | Homo sapiens | |||
8. | ALA4064397 | 16 | Efficacy | = | -2.2 | % | ALA4028339 | % | Homo sapiens | |||
9. | ALA4064397 | 16 | Efficacy | = | -4.2 | % | ALA4028340 | % | Homo sapiens | |||
10. | ALA4064397 | 16 | Efficacy | = | 0.5 | % | ALA4028341 | % | Homo sapiens | |||
11. | ALA4064397 | 16 | Efficacy | = | -2.8 | % | ALA4028342 | % | Homo sapiens | |||
12. | ALA4064397 | 16 | Efficacy | = | 0.3 | % | ALA4028343 | % | Homo sapiens | |||
13. | ALA4064397 | 16 | Efficacy | = | 0.5 | % | ALA4028344 | % | Homo sapiens | |||
14. | ALA4064397 | 16 | Efficacy | = | -7.6 | % | ALA4028345 | % | Homo sapiens | |||
15. | ALA4064397 | 16 | Efficacy | = | 73.4 | % | ALA4028346 | % | Homo sapiens | |||
16. | ALA4064397 | 16 | Efficacy | = | -11 | % | ALA4028347 | % | Homo sapiens | |||
17. | ALA4064397 | 16 | Efficacy | = | -3.9 | % | ALA4028348 | % | Homo sapiens | |||
18. | ALA4064397 | 16 | EC50 | = | 13.7 | nM | ALA4028349 | 7.86 | nM | Homo sapiens | ||
19. | ALA4064397 | 16 | CC50 | > | 100 | uM | ALA4028350 | nM | Homo sapiens | |||
20. | ALA4064397 | 16 | Cmax | = | 16400 | ng/ml | ALA4028351 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Mus musculus |