# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4065412 | 35 | Activity | = | 39 | % | ALA4019765 | % | Homo sapiens | |||
2. | ALA4065412 | 35 | IC50 | = | 24 | nM | ALA4019776 | 7.62 | nM | Homo sapiens | ||
3. | ALA4065412 | 35 | CL | = | 6173 | ml/hr/kg | ALA4019775 | mL.min-1.kg-1 | Rattus norvegicus | |||
4. | ALA4065412 | 35 | Vdss | = | 6229 | ml/kg | ALA4019774 | L.kg-1 | Rattus norvegicus | |||
5. | ALA4065412 | 35 | Cmax | = | 745 | ng/ml | ALA4019773 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
6. | ALA4065412 | 35 | beta t1/2 | = | 1.8 | hr | ALA4019772 | hr | Rattus norvegicus | |||
7. | ALA4065412 | 35 | TGI | = | 69 | % | ALA4019770 | % | Homo sapiens | |||
8. | ALA4065412 | 35 | deltaTm | = | 1.58 | degrees C | ALA4019769 | degrees C | Homo sapiens | |||
9. | ALA4065412 | 35 | INH | 0 | ALA4019768 | Active | % | Homo sapiens | ||||
10. | ALA4065412 | 35 | INH | 0 | ALA4019767 | Active | % | |||||
11. | ALA4065412 | 35 | INH | 0 | ALA4019766 | Active | % | |||||
12. | ALA4065412 | 35 | Activity | = | 19 | % | ALA4019764 | % | Homo sapiens | |||
13. | ALA4065412 | 35 | Activity | 0 | ALA4019763 | Active | Homo sapiens | |||||
14. | ALA4065412 | 35 | Activity | 0 | ALA4019762 | Not Active | Homo sapiens | |||||
15. | ALA4065412 | 35 | Activity | 0 | ALA4019761 | Active | Homo sapiens | |||||
16. | ALA4065412 | 35 | Activity | = | 2.19 | % | ALA4019760 | % | Homo sapiens | |||
17. | ALA4065412 | 35 | Activity | = | 15.22 | % | ALA4019759 | % | Homo sapiens | |||
18. | ALA4065412 | 35 | Activity | = | 12.46 | % | ALA4019758 | % | Homo sapiens | |||
19. | ALA4065412 | 35 | Activity | = | 2.43 | % | ALA4019757 | % | Homo sapiens | |||
20. | ALA4065412 | 35 | Activity | = | 21.84 | % | ALA4019756 | % | Homo sapiens |