# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4065603 | LSPN423, diastereomeric mixture 69:31 | IC50 | = | 11.51 | uM | ALA4044524 | 4.94 | nM | Homo sapiens | ||
2. | ALA4065603 | LSPN423, diastereomeric mixture 69:31 | IC50 | = | 11.12 | uM | ALA4044525 | 4.95 | nM | Homo sapiens | ||
3. | ALA4065603 | LSPN423, diastereomeric mixture 69:31 | IC50 | = | 9.78 | uM | ALA4044526 | 5.01 | nM | Homo sapiens | ||
4. | ALA4065603 | LSPN423, diastereomeric mixture 69:31 | IC50 | = | 5.13 | uM | ALA4044527 | 5.29 | nM | Homo sapiens | ||
5. | ALA4065603 | LSPN423, diastereomeric mixture 69:31 | IC50 | = | 5.26 | uM | ALA4044528 | 5.28 | nM | Homo sapiens | ||
6. | ALA4065603 | LSPN423, diastereomeric mixture 69:31 | IC50 | = | 7.17 | uM | ALA4044529 | 5.14 | nM | Homo sapiens | ||
7. | ALA4065603 | LSPN423, diastereomeric mixture 69:31 | IC50 | = | 5.75 | uM | ALA4044530 | 5.24 | nM | Homo sapiens | ||
8. | ALA4065603 | LSPN423, diastereomeric mixture 69:31 | IC50 | = | 6.09 | uM | ALA4044531 | 5.21 | nM | Homo sapiens | ||
9. | ALA4065603 | LSPN423, diastereomeric mixture 69:31 | INH | = | 98.5 | % | ALA4044516 | % | Homo sapiens | |||
10. | ALA4065603 | LSPN423, diastereomeric mixture 69:31 | IC50 | = | 16.86 | uM | ALA4044523 | 4.77 | nM | Homo sapiens | ||
11. | ALA4065603 | LSPN423, diastereomeric mixture 69:31 | Ki | = | 1.33 | uM | ALA4044522 | 5.88 | nM | Homo sapiens | ||
12. | ALA4065603 | LSPN423, diastereomeric mixture 69:31 | INH | 0 | ALA4044521 | Active | % | Homo sapiens | ||||
13. | ALA4065603 | LSPN423, diastereomeric mixture 69:31 | IC50 | = | 5.72 | uM | ALA4044519 | 5.24 | nM | Homo sapiens | ||
14. | ALA4065603 | LSPN423, diastereomeric mixture 69:31 | INH | = | 30.8 | % | ALA4044518 | % | Homo sapiens | |||
15. | ALA4065603 | LSPN423, diastereomeric mixture 69:31 | INH | = | 78 | % | ALA4044517 | % | Homo sapiens | |||
16. | ALA4065603 | LSPN423, diastereomeric mixture 69:31 | IC50 | = | 5.36 | uM | ALA4625550 | 5.27 | nM | Homo sapiens | ||
17. | ALA4065603 | LSPN423, diastereomeric mixture 69:31 | IC50 | = | 5.72 | uM | ALA4625549 | 5.24 | nM | Homo sapiens |