| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4065973 | 11 | Time | = | 60 | min | ALA5233312 | hr | Mus musculus | |||
| 2. | ALA4065973 | 11 | Activity | = | 31.98 | mmHg | ALA5233311 | mmHg | Mus musculus | |||
| 3. | ALA4065973 | 11 | pEC50 | = | 8.56 | ALA5233310 | 8.56 | nM | Homo sapiens | |||
| 4. | ALA4065973 | 11 | pKi | = | 9.35 | ALA5233309 | 9.35 | nM | Rattus norvegicus | |||
| 5. | ALA4065973 | 11 | PPB | = | 55 | % | ALA5233308 | % | ||||
| 6. | ALA4065973 | 11 | t1/2 | = | 0.99 | hr | ALA5233307 | hr | ||||
| 7. | ALA4065973 | 11 | t1/2 | = | 8.29 | hr | ALA5233306 | hr | ||||
| 8. | ALA4065973 | 11 | t1/2 | > | 48 | hr | ALA5233304 | hr | Homo sapiens | |||
| 9. | ALA4065973 | 11 | EC50 | = | 4.9 | nM | ALA4401048 | 8.31 | nM | Homo sapiens | ||
| 10. | ALA4065973 | 11 | Activity | = | -36 | mmHg | ALA4401049 | mmHg | Mus musculus | |||
| 11. | ALA4065973 | 11 | Activity | 0 | ALA4401049 | Tde | Mus musculus | |||||
| 12. | ALA4065973 | 11 | Km | = | 245 | uM | ALA4401034 | nM | Homo sapiens | |||
| 13. | ALA4065973 | 11 | Kcat | = | 16.5 | /s | ALA4401035 | /s | Homo sapiens | |||
| 14. | ALA4065973 | 11 | Kcat/Km | = | 6.7 | 10'4/Ms | ALA4401036 | 10'4/Ms | Homo sapiens | |||
| 15. | ALA4065973 | 11 | Vmax | = | 3.706 | micromol/min | ALA4401043 | micromol/min | Homo sapiens | |||
| 16. | ALA4065973 | 11 | t1/2 | > | 30 | hr | ALA4401044 | hr | Homo sapiens | |||
| 17. | ALA4065973 | 11 | t1/2 | = | 0.9 | hr | ALA4401045 | hr | Homo sapiens | |||
| 18. | ALA4065973 | 11 | t1/2 | = | 1.2 | hr | ALA4401046 | hr | Homo sapiens | |||
| 19. | ALA4065973 | 11 | INH | 0 | ALA4401047 | Active | % | Rattus norvegicus | ||||
| 20. | ALA4065973 | 11 | FC | = | 778 | ALA4703010 | Mus musculus |
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