# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4066040 | 12 | % of inhibition | = | 63.5 | % | ALA5214502 | % | Homo sapiens | |||
2. | ALA4066040 | 12 | % of inhibition | = | 63.9 | % | ALA5214500 | % | Homo sapiens | |||
3. | ALA4066040 | 12 | Ki | = | 1192.34 | nM | ALA5214507 | 5.92 | nM | Homo sapiens | ||
4. | ALA4066040 | 12 | Ki | = | 314.63 | nM | ALA5214505 | 6.50 | nM | Homo sapiens | ||
5. | ALA4066040 | 12 | % of control | = | 51 | % | ALA5214503 | % | Homo sapiens | |||
6. | ALA4066040 | 12 | Ki | = | 19.59 | nM | ALA5214506 | 7.71 | nM | Homo sapiens | ||
7. | ALA4066040 | 12 | EC50 | = | 130 | nM | ALA5214504 | 6.89 | nM | Homo sapiens | ||
8. | ALA4066040 | 12 | % of inhibition | = | 95.5 | % | ALA5214508 | % | Homo sapiens | |||
9. | ALA4066040 | 12 | % of inhibition | = | 63.5 | % | ALA5214501 | % | Homo sapiens | |||
10. | ALA4066040 | 12 | % of inhibition | = | 63.9 | % | ALA5214499 | % | Homo sapiens | |||
11. | ALA4066040 | 12 | EC50 | = | 28 | nM | ALA5210279 | 7.55 | nM | Homo sapiens | ||
12. | ALA4066040 | 12 | EC50 | = | 35 | nM | ALA5210086 | 7.46 | nM | Homo sapiens | ||
13. | ALA4066040 | 12 | CL free | = | 775 | L/hr/kg | ALA4022902 | mL.min-1.kg-1 | ||||
14. | ALA4066040 | 12 | CL free | = | 1250 | L/hr/kg | ALA4022901 | mL.min-1.kg-1 | ||||
15. | ALA4066040 | 12 | permeability | = | 0.3 | 10'-6 cm/s | ALA4022900 | 10'-6 cm/s | ||||
16. | ALA4066040 | 12 | Activity | < | 30 | % | ALA4022899 | % | Homo sapiens | |||
17. | ALA4066040 | 12 | EC50 | = | 1 | uM | ALA4022894 | 6.00 | nM | Homo sapiens | ||
18. | ALA4066040 | 12 | max activation | = | 69 | % | ALA4022895 | % | Homo sapiens | |||
19. | ALA4066040 | 12 | logD | = | 4.96 | ALA4022896 | ||||||
20. | ALA4066040 | 12 | Growth Rate | = | 1 | ALA4725213 | Homo sapiens |