# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4066104 | 41; CHMFL-BMX-078 | Activity | 0 | ALA4008372 | Active | Homo sapiens | |||||
2. | ALA4066104 | 41; CHMFL-BMX-078 | Cmax | = | 5.58 | ng/ml | ALA4008370 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
3. | ALA4066104 | 41; CHMFL-BMX-078 | Cmax | = | 13565.23 | ng/ml | ALA4008369 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
4. | ALA4066104 | 41; CHMFL-BMX-078 | Tmax | = | 0.19 | hr | ALA4008368 | hr | Rattus norvegicus | |||
5. | ALA4066104 | 41; CHMFL-BMX-078 | Tmax | = | 0.017 | hr | ALA4008367 | hr | Rattus norvegicus | |||
6. | ALA4066104 | 41; CHMFL-BMX-078 | t1/2 | = | 6.11 | hr | ALA4008366 | hr | Rattus norvegicus | |||
7. | ALA4066104 | 41; CHMFL-BMX-078 | t1/2 | = | 0.8 | hr | ALA4008365 | hr | Rattus norvegicus | |||
8. | ALA4066104 | 41; CHMFL-BMX-078 | MRT(t) | = | 2.76 | hr | ALA4008364 | hr | Rattus norvegicus | |||
9. | ALA4066104 | 41; CHMFL-BMX-078 | MRT(t) | = | 0.224 | hr | ALA4008363 | hr | Rattus norvegicus | |||
10. | ALA4066104 | 41; CHMFL-BMX-078 | AUC | = | 27.63 | ng/mL.hr | ALA4008362 | ng.hr.mL-1 | Rattus norvegicus | |||
11. | ALA4066104 | 41; CHMFL-BMX-078 | AUC | = | 1388.25 | ng/mL.hr | ALA4008361 | ng.hr.mL-1 | Rattus norvegicus | |||
12. | ALA4066104 | 41; CHMFL-BMX-078 | AUCt | = | 13.39 | ng/mL.hr | ALA4008360 | ng.hr.mL-1 | Rattus norvegicus | |||
13. | ALA4066104 | 41; CHMFL-BMX-078 | AUCt | = | 1386.41 | ng/mL.hr | ALA4008359 | ng.hr.mL-1 | Rattus norvegicus | |||
14. | ALA4066104 | 41; CHMFL-BMX-078 | INH | 0 | ALA4008358 | Active | % | Homo sapiens | ||||
15. | ALA4066104 | 41; CHMFL-BMX-078 | GI50 | > | 10 | uM | ALA4008354 | nM | Cricetulus griseus | |||
16. | ALA4066104 | 41; CHMFL-BMX-078 | GI50 | > | 10 | uM | ALA4008348 | nM | ||||
17. | ALA4066104 | 41; CHMFL-BMX-078 | GI50 | = | 4.93 | uM | ALA4008357 | nM | Homo sapiens | |||
18. | ALA4066104 | 41; CHMFL-BMX-078 | GI50 | > | 10 | uM | ALA4008356 | nM | Homo sapiens | |||
19. | ALA4066104 | 41; CHMFL-BMX-078 | GI50 | > | 10 | uM | ALA4008353 | nM | Homo sapiens | |||
20. | ALA4066104 | 41; CHMFL-BMX-078 | GI50 | > | 10 | uM | ALA4008352 | nM | Homo sapiens |