# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4066494 | 1; A-705253 | Drug metabolism | 0 | ALA4041074 | Metabolite_Notdetected | ||||||
2. | ALA4066494 | 1; A-705253 | INH | 0 | ALA4041073 | Active | % | Homo sapiens | ||||
3. | ALA4066494 | 1; A-705253 | INH | = | 84 | % | ALA4041067 | % | Homo sapiens | |||
4. | ALA4066494 | 1; A-705253 | INH | = | 94 | % | ALA4041066 | % | Homo sapiens | |||
5. | ALA4066494 | 1; A-705253 | Ki | = | 1.8 | nM | ALA4041065 | 8.74 | nM | Homo sapiens | ||
6. | ALA4066494 | 1; A-705253 | Ki | = | 28 | nM | ALA4041064 | 7.55 | nM | Homo sapiens | ||
7. | ALA4066494 | 1; A-705253 | Ki | = | 3290 | nM | ALA4041063 | 5.48 | nM | Homo sapiens | ||
8. | ALA4066494 | 1; A-705253 | Ki | = | 137 | nM | ALA4040999 | 6.86 | nM | |||
9. | ALA4066494 | 1; A-705253 | Ratio Ki | = | 59 | ALA4041007 | ||||||
10. | ALA4066494 | 1; A-705253 | Ratio Ki | = | 2.5 | ALA4041006 | ||||||
11. | ALA4066494 | 1; A-705253 | Ratio Ki | < | 0.1 | ALA4041005 | ||||||
12. | ALA4066494 | 1; A-705253 | Ratio Ki | < | 1 | ALA4041004 | ||||||
13. | ALA4066494 | 1; A-705253 | Ki | = | 56 | nM | ALA4041003 | 7.25 | nM | Homo sapiens |