| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4067502 | 15 | EC50 | > | 10000 | nM | ALA4051064 | nM | Homo sapiens | |||
| 2. | ALA4067502 | 15 | EC50 | > | 10000 | nM | ALA4051065 | nM | Homo sapiens | |||
| 3. | ALA4067502 | 15 | EC50 | = | 18 | nM | ALA4051035 | 7.75 | nM | Homo sapiens | ||
| 4. | ALA4067502 | 15 | Intrinsic activity | = | 105 | % | ALA4051036 | % | Homo sapiens | |||
| 5. | ALA4067502 | 15 | EC50 | > | 10000 | nM | ALA4051037 | nM | Homo sapiens | |||
| 6. | ALA4067502 | 15 | Intrinsic activity | = | 0 | % | ALA4051038 | % | Homo sapiens | |||
| 7. | ALA4067502 | 15 | Ratio EC50 | > | 556 | ALA4051039 | ||||||
| 8. | ALA4067502 | 15 | CLH | = | 57 | ml/min.kg | ALA4051040 | mL.min-1.kg-1 | Homo sapiens | |||
| 9. | ALA4067502 | 15 | INH | < | 34 | % | ALA4051055 | % | Homo sapiens | |||
| 10. | ALA4067502 | 15 | INH | < | 34 | % | ALA4051056 | % | Homo sapiens | |||
| 11. | ALA4067502 | 15 | INH | < | 34 | % | ALA4051057 | % | Homo sapiens | |||
| 12. | ALA4067502 | 15 | INH | < | 34 | % | ALA4051058 | % | Homo sapiens | |||
| 13. | ALA4067502 | 15 | Activity | = | 5.8 | % | ALA4051059 | % | Rattus norvegicus | |||
| 14. | ALA4067502 | 15 | Activity | = | 0.9 | % | ALA4051060 | % | Rattus norvegicus | |||
| 15. | ALA4067502 | 15 | Activity | = | 2 | % | ALA4051061 | % | Rattus norvegicus | |||
| 16. | ALA4067502 | 15 | Activity | = | 12.9 | % | ALA4051062 | % | Rattus norvegicus | |||
| 17. | ALA4067502 | 15 | Activity | 0 | ALA4051063 | Dose-dependent effect | Callithrix jacchus | |||||
| 18. | ALA4067502 | 15 | permeability | = | 5 | 10'-6 cm/s | ALA4051047 | 10'-6 cm/s | ||||
| 19. | ALA4067502 | 15 | Intrinsic activity | = | 4 | % | ALA4051051 | % | Homo sapiens | |||
| 20. | ALA4067502 | 15 | INH | < | 34 | % | ALA4051054 | % | Homo sapiens |
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