# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4067973 | 6 | pKi | = | 7.05 | ALA4416333 | 7.05 | nM | Homo sapiens | |||
2. | ALA4067973 | 6 | Activity | 0 | ALA4306974 | Not Active | Homo sapiens | |||||
3. | ALA4067973 | 6 | IC50 | = | 4.36 | uM | ALA4306964 | 5.36 | nM | Homo sapiens | ||
4. | ALA4067973 | 6 | INH | >= | 50 | % | ALA4306965 | % | Homo sapiens | |||
5. | ALA4067973 | 6 | deltaS | = | 10 | cal/mol/deg | ALA4028407 | cal/mol/deg | Homo sapiens | |||
6. | ALA4067973 | 6 | deltaH | = | -4600 | cal/mol | ALA4028406 | cal/mol | Homo sapiens | |||
7. | ALA4067973 | 6 | INH | 0 | ALA4028405 | Active | % | Homo sapiens | ||||
8. | ALA4067973 | 6 | INH | 0 | ALA4028404 | Active | % | Homo sapiens | ||||
9. | ALA4067973 | 6 | IC50 | = | 62 | uM | ALA4028403 | 4.21 | nM | Homo sapiens | ||
10. | ALA4067973 | 6 | IC50 | = | 40 | uM | ALA4028402 | 4.40 | nM | Homo sapiens | ||
11. | ALA4067973 | 6 | IC50 | = | 20 | uM | ALA4028401 | 4.70 | nM | Homo sapiens | ||
12. | ALA4067973 | 6 | IC50 | = | 1.3 | uM | ALA4028400 | 5.89 | nM | Homo sapiens | ||
13. | ALA4067973 | 6 | Kd | = | 2.7 | uM | ALA4028399 | 5.57 | nM | Homo sapiens | ||
14. | ALA4067973 | 6 | IC50 | = | 14 | uM | ALA4028398 | 4.85 | nM | Homo sapiens |