# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4069833 | 9 | IC50 | = | 839.7 | nM | ALA4029859 | 6.08 | nM | Homo sapiens | ||
2. | ALA4069833 | 9 | Drug uptake | = | 9.22 | nM | ALA4029896 | nM | ||||
3. | ALA4069833 | 9 | Cp | = | 7.5 | uM | ALA4029895 | uM | ||||
4. | ALA4069833 | 9 | INH | 0 | ALA4029891 | Not Active | % | Homo sapiens | ||||
5. | ALA4069833 | 9 | INH | 0 | ALA4029890 | Not Active | % | Homo sapiens | ||||
6. | ALA4069833 | 9 | INH | 0 | ALA4029889 | Not Active | % | Homo sapiens | ||||
7. | ALA4069833 | 9 | INH | 0 | ALA4029888 | Not Active | % | Homo sapiens | ||||
8. | ALA4069833 | 9 | INH | 0 | ALA4029882 | Not Active | % | Homo sapiens | ||||
9. | ALA4069833 | 9 | INH | = | 38 | % | ALA4029892 | % | Cavia porcellus | |||
10. | ALA4069833 | 9 | INH | = | 27.2 | % | ALA4029887 | % | Homo sapiens | |||
11. | ALA4069833 | 9 | Ratio IC50 | > | 70 | ALA4029886 | ||||||
12. | ALA4069833 | 9 | Ratio IC50 | > | 200 | ALA4029885 | ||||||
13. | ALA4069833 | 9 | INH | = | 24.21 | % | ALA4029884 | % | Homo sapiens | |||
14. | ALA4069833 | 9 | INH | = | 2.37 | % | ALA4029883 | % | Homo sapiens | |||
15. | ALA4069833 | 9 | Tmax | = | 24 | hr | ALA4029881 | hr | Cavia porcellus | |||
16. | ALA4069833 | 9 | AUC | = | 13427 | ng.hr/ml | ALA4029880 | ng.hr.mL-1 | Cavia porcellus | |||
17. | ALA4069833 | 9 | Cmax | = | 803 | ng/ml | ALA4029879 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Cavia porcellus | ||
18. | ALA4069833 | 9 | t1/2 | = | 11.2 | hr | ALA4029878 | hr | Rattus norvegicus | |||
19. | ALA4069833 | 9 | F | = | 33 | % | ALA4029877 | % | Rattus norvegicus | |||
20. | ALA4069833 | 9 | Tmax | = | 4 | hr | ALA4029876 | hr | Rattus norvegicus |