| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4071576 | 35 | t1/2 | = | 37 | min | ALA4324314 | hr | Homo sapiens | |||
| 2. | ALA4071576 | 35 | t1/2 | = | 11.9 | min | ALA4324313 | hr | Homo sapiens | |||
| 3. | ALA4071576 | 35 | Kdiss | = | 3.2 | 10'-4/s | ALA4324312 | 10'-4/s | Homo sapiens | |||
| 4. | ALA4071576 | 35 | Kdiss | = | 1 | 10'-3/s | ALA4324311 | 10'-3/s | Homo sapiens | |||
| 5. | ALA4071576 | 35 | Ka | = | 1.9 | 10'-6/M/s | ALA4324310 | 10'-6/M/s | Homo sapiens | |||
| 6. | ALA4071576 | 35 | Ka | = | 1.3 | 10'-6/M/s | ALA4324309 | 10'-6/M/s | Homo sapiens | |||
| 7. | ALA4071576 | 35 | pKd | = | 9.8 | ALA4324308 | 9.80 | nM | Homo sapiens | |||
| 8. | ALA4071576 | 35 | pKd | = | 9.1 | ALA4324307 | 9.10 | nM | Homo sapiens | |||
| 9. | ALA4071576 | 35 | solubility | > | 480 | uM | ALA4324289 | nM | ||||
| 10. | ALA4071576 | 35 | logD | = | 2.5 | ALA4324288 | ||||||
| 11. | ALA4071576 | 35 | IC50 | = | 0.062 | uM | ALA4324287 | 7.21 | nM | Homo sapiens | ||
| 12. | ALA4071576 | 35 | IC50 | = | 0.012 | uM | ALA4324286 | 7.92 | nM | Homo sapiens | ||
| 13. | ALA4071576 | 35 | IC50 | = | 0.001 | uM | ALA4324285 | 9.30 | nM | Homo sapiens | ||
| 14. | ALA4071576 | 35 | IC50 | < | 0 | uM | ALA4324284 | nM | Homo sapiens | |||
| 15. | ALA4071576 | 35 | Ratio | = | 9.6 | ALA4051381 | ||||||
| 16. | ALA4071576 | 35 | Papp | = | 52 | ucm/s | ALA4051380 | ucm/s | ||||
| 17. | ALA4071576 | 35 | Activity | 0 | ALA4051379 | Active | Homo sapiens | |||||
| 18. | ALA4071576 | 35 | Activity | 0 | ALA4051378 | Active | Mus musculus | |||||
| 19. | ALA4071576 | 35 | F | = | 87 | % | ALA4051377 | % | Canis lupus familiaris | |||
| 20. | ALA4071576 | 35 | Vdss | = | 0.9 | L/Kg | ALA4051376 | L.kg-1 | Canis lupus familiaris |
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