| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4071600 | 19 | solubility | > | 1000 | ug ml-1 | ALA4047179 | ug.mL-1 | ||||
| 2. | ALA4071600 | 19 | solubility | > | 1000 | ug ml-1 | ALA4047178 | ug.mL-1 | ||||
| 3. | ALA4071600 | 19 | solubility | > | 1000 | ug ml-1 | ALA4047177 | ug.mL-1 | ||||
| 4. | ALA4071600 | 19 | %max | = | 62 | % | ALA4047163 | % | Mus musculus | |||
| 5. | ALA4071600 | 19 | pEC50 | = | 6.6 | ALA4047163 | 6.60 | nM | Mus musculus | |||
| 6. | ALA4071600 | 19 | %max | = | 66 | % | ALA4047176 | % | Rattus norvegicus | |||
| 7. | ALA4071600 | 19 | pEC50 | = | 6.5 | ALA4047176 | 6.50 | nM | Rattus norvegicus | |||
| 8. | ALA4071600 | 19 | fCmax | = | 3 | ng/ml | ALA4047175 | ng/ml | Rattus norvegicus | |||
| 9. | ALA4071600 | 19 | fCmax | = | 7 | nM | ALA4047174 | nM | Rattus norvegicus | |||
| 10. | ALA4071600 | 19 | PPB | = | 93 | % | ALA4047173 | % | Rattus norvegicus | |||
| 11. | ALA4071600 | 19 | AUC | = | 266 | hr.ng/ml | ALA4047172 | ng.hr.mL-1 | Rattus norvegicus | |||
| 12. | ALA4071600 | 19 | AUC | = | 265 | hr.ng/ml | ALA4047171 | ng.hr.mL-1 | Rattus norvegicus | |||
| 13. | ALA4071600 | 19 | Drug recovery | = | 86.3 | % | ALA4047170 | % | ||||
| 14. | ALA4071600 | 19 | Cmax | = | 48 | ng/ml | ALA4047168 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 15. | ALA4071600 | 19 | Cmax | = | 57 | ng/ml | ALA4047166 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 16. | ALA4071600 | 19 | t1/2 | > | 12 | hr | ALA4047165 | hr | ||||
| 17. | ALA4071600 | 19 | Papp | = | 3 | nm/s | ALA4047164 | nm/s | ||||
| 18. | ALA4071600 | 19 | pEC50 | = | 7.3 | ALA4047162 | 7.30 | nM | Homo sapiens | |||
| 19. | ALA4071600 | 19 | EC50 | = | 50 | nM | ALA4047162 | 7.30 | nM | Homo sapiens | ||
| 20. | ALA4071600 | 19 | %max | = | 84 | % | ALA4047162 | % | Homo sapiens |
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