# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4073780 | 21 | BPR | = | 1.4 | ALA4040868 | ||||||
2. | ALA4073780 | 21 | BPR | = | 1.9 | ALA4040867 | ||||||
3. | ALA4073780 | 21 | F | = | 26 | % | ALA4040866 | % | Mus musculus | |||
4. | ALA4073780 | 21 | F | = | 56 | % | ALA4040865 | % | Rattus norvegicus | |||
5. | ALA4073780 | 21 | CL | = | 2.6 | L/hr/kg | ALA4040864 | mL.min-1.kg-1 | Mus musculus | |||
6. | ALA4073780 | 21 | CL | = | 1.5 | L/hr/kg | ALA4040863 | mL.min-1.kg-1 | Rattus norvegicus | |||
7. | ALA4073780 | 21 | CLH | = | 5 | L/hr/kg | ALA4040862 | mL.min-1.kg-1 | ||||
8. | ALA4073780 | 21 | CLH | = | 2.5 | L/hr/kg | ALA4040861 | mL.min-1.kg-1 | ||||
9. | ALA4073780 | 21 | CLH | = | 0.3 | L/hr/kg | ALA4040860 | mL.min-1.kg-1 | ||||
10. | ALA4073780 | 21 | Therm_solubility | = | 1.9 | uM | ALA4040859 | nM | ||||
11. | ALA4073780 | 21 | logD | = | 4.6 | ALA4040858 | ||||||
12. | ALA4073780 | 21 | Emax | = | 330 | % | ALA4040857 | % | Homo sapiens | |||
13. | ALA4073780 | 21 | EC50 | = | 110 | nM | ALA4040856 | 6.96 | nM | Homo sapiens | ||
14. | ALA4073780 | 21 | Emax | = | 725 | % | ALA4040855 | % | Homo sapiens | |||
15. | ALA4073780 | 21 | EC50 | = | 225 | nM | ALA4040854 | 6.65 | nM | Homo sapiens | ||
16. | ALA4073780 | 21 | IC50 | = | 13 | nM | ALA4040853 | 7.89 | nM |