# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4075458 | 6a | Activity | 0 | ALA4059060 | Not Active | Homo sapiens | |||||
2. | ALA4075458 | 6a | Activity | 0 | ALA4059059 | Active | Homo sapiens | |||||
3. | ALA4075458 | 6a | Activity | 0 | ALA4059058 | Not Active | Homo sapiens | |||||
4. | ALA4075458 | 6a | Activity | 0 | ALA4059057 | Not Active | Homo sapiens | |||||
5. | ALA4075458 | 6a | INH | 0 | ALA4059056 | Active | % | Homo sapiens | ||||
6. | ALA4075458 | 6a | INH | 0 | ALA4059055 | Active | % | Homo sapiens | ||||
7. | ALA4075458 | 6a | INH | 0 | ALA4059054 | Active | % | Homo sapiens | ||||
8. | ALA4075458 | 6a | INH | 0 | ALA4059053 | Active | % | Homo sapiens | ||||
9. | ALA4075458 | 6a | INH | 0 | ALA4059052 | Active | % | Homo sapiens | ||||
10. | ALA4075458 | 6a | INH | 0 | ALA4059051 | Active | % | Homo sapiens | ||||
11. | ALA4075458 | 6a | Activity | 0 | ALA4059044 | Dose-dependent effect | Homo sapiens | |||||
12. | ALA4075458 | 6a | INH | 0 | ALA4059050 | Not Active | % | Homo sapiens | ||||
13. | ALA4075458 | 6a | INH | 0 | ALA4059045 | Active | % | Homo sapiens | ||||
14. | ALA4075458 | 6a | Activity | 0 | ALA4059049 | Not Active | ||||||
15. | ALA4075458 | 6a | Activity | 0 | ALA4059048 | Not Active | ||||||
16. | ALA4075458 | 6a | Kd | = | 4.5 | uM | ALA4059044 | 5.35 | nM | Homo sapiens | ||
17. | ALA4075458 | 6a | Activity | 0 | ALA4059066 | Active | Homo sapiens | |||||
18. | ALA4075458 | 6a | Activity | 0 | ALA4059065 | Active | Homo sapiens | |||||
19. | ALA4075458 | 6a | IC50 | = | 26.47 | uM | ALA4059064 | 4.58 | nM | Homo sapiens | ||
20. | ALA4075458 | 6a | IC50 | = | 24.17 | uM | ALA4059063 | 4.62 | nM | Homo sapiens |