# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4076839 | trans-(+)-1d | Ki | = | 7 | nM | ALA4033549 | 8.15 | nM | Cavia porcellus | ||
2. | ALA4076839 | trans-(+)-1d | Ki | = | 1837 | nM | ALA4033550 | 5.74 | nM | |||
3. | ALA4076839 | trans-(+)-1d | K | = | 0.51 | /hr | ALA4033561 | /hr | Mus musculus | |||
4. | ALA4076839 | trans-(+)-1d | t1/2 | = | 65.2 | hr | ALA4033562 | hr | Homo sapiens | |||
5. | ALA4076839 | trans-(+)-1d | K | = | 0.01 | /hr | ALA4033563 | /hr | Homo sapiens | |||
6. | ALA4076839 | trans-(+)-1d | Activity | 0 | ALA4033564 | Not Active | Mus musculus | |||||
7. | ALA4076839 | trans-(+)-1d | Activity | 0 | ALA4033571 | Not Active | Rattus norvegicus | |||||
8. | ALA4076839 | trans-(+)-1d | Activity | 0 | ALA4033572 | Not Active | ||||||
9. | ALA4076839 | trans-(+)-1d | Activity | 0 | ALA4033573 | Not Active | Rattus norvegicus | |||||
10. | ALA4076839 | trans-(+)-1d | Activity | 0 | ALA4033574 | Not Active | Rattus norvegicus | |||||
11. | ALA4076839 | trans-(+)-1d | Activity | 0 | ALA4033575 | Not Active | Rattus norvegicus | |||||
12. | ALA4076839 | trans-(+)-1d | Activity | 0 | ALA4033577 | Active | Mus musculus | |||||
13. | ALA4076839 | trans-(+)-1d | solubility | = | 3.1 | mg/ml | ALA4033554 | ug.mL-1 | ||||
14. | ALA4076839 | trans-(+)-1d | Ratio Ki | > | 250 | ALA4033553 | ||||||
15. | ALA4076839 | trans-(+)-1d | t1/2 | = | 1.14 | hr | ALA4033560 | hr | Mus musculus | |||
16. | ALA4076839 | trans-(+)-1d | K | = | 3.26 | /hr | ALA4033548 | /hr | Rattus norvegicus | |||
17. | ALA4076839 | trans-(+)-1d | t1/2 | = | 0.38 | hr | ALA4033559 | hr | Rattus norvegicus | |||
18. | ALA4076839 | trans-(+)-1d | K | = | 0.009 | /hr | ALA4033558 | /hr | ||||
19. | ALA4076839 | trans-(+)-1d | K | = | 0.009 | /hr | ALA4033557 | /hr | ||||
20. | ALA4076839 | trans-(+)-1d | t1/2 | = | 91 | hr | ALA4033556 | hr |