# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4077061 | 24 | Ratio | = | 2.5 | ALA4010347 | ||||||
2. | ALA4077061 | 24 | Stability | > | 115 | min | ALA4010346 | min | Homo sapiens | |||
3. | ALA4077061 | 24 | Activity | 0 | ALA4010345 | Active | Mus musculus | |||||
4. | ALA4077061 | 24 | Fu | = | 47 | nM | ALA4010344 | nM | ||||
5. | ALA4077061 | 24 | Fu | = | 63 | nM | ALA4010343 | nM | Mus musculus | |||
6. | ALA4077061 | 24 | Cp(f) | = | 173 | nM | ALA4010342 | nM | Mus musculus | |||
7. | ALA4077061 | 24 | logD | = | 1.9 | ALA4010341 | ||||||
8. | ALA4077061 | 24 | Kinetic_solubility | = | 31 | uM | ALA4010340 | nM | ||||
9. | ALA4077061 | 24 | Ratio | = | 2.3 | ALA4010339 | ||||||
10. | ALA4077061 | 24 | Papp | = | 13 | 10'-6 cm/s | ALA4010338 | 10'-6 cm/s | ||||
11. | ALA4077061 | 24 | CLH(app) | < | 8.4 | uL/min.mg | ALA4010337 | mL.min-1.g-1 | Homo sapiens | |||
12. | ALA4077061 | 24 | IC50 | = | 52 | uM | ALA4010336 | 4.28 | nM | Homo sapiens | ||
13. | ALA4077061 | 24 | IC50 | = | 0.11 | nM | ALA4010335 | 9.96 | nM | Homo sapiens |