# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4078272 | 3-(S) | IP | = | 1729 | nM | ALA4012173 | nM | ||||
2. | ALA4078272 | 3-(S) | Ratio | = | 16 | ALA4012178 | ||||||
3. | ALA4078272 | 3-(S) | Ratio | = | 3 | ALA4012177 | ||||||
4. | ALA4078272 | 3-(S) | Ratio | = | 9 | ALA4012176 | ||||||
5. | ALA4078272 | 3-(S) | Ratio | = | 11 | ALA4012175 | ||||||
6. | ALA4078272 | 3-(S) | Ratio | = | 2 | ALA4012174 | ||||||
7. | ALA4078272 | 3-(S) | Ratio | = | 1 | ALA4012162 | ||||||
8. | ALA4078272 | 3-(S) | IP | = | 1545 | nM | ALA4012172 | nM | Human immunodeficiency virus 1 | |||
9. | ALA4078272 | 3-(S) | IP | = | 271 | nM | ALA4012171 | nM | Human immunodeficiency virus 1 | |||
10. | ALA4078272 | 3-(S) | IP | = | 820 | nM | ALA4012170 | nM | Human immunodeficiency virus 1 | |||
11. | ALA4078272 | 3-(S) | IP | = | 1006 | nM | ALA4012169 | nM | Human immunodeficiency virus 1 | |||
12. | ALA4078272 | 3-(S) | IP | = | 142 | nM | ALA4012168 | nM | Human immunodeficiency virus 1 | |||
13. | ALA4078272 | 3-(S) | IP | = | 123 | nM | ALA4012167 | nM | Human immunodeficiency virus 1 | |||
14. | ALA4078272 | 3-(S) | IP | = | 95 | nM | ALA4012166 | nM | ||||
15. | ALA4078272 | 3-(S) | F | = | 44 | % | ALA4012164 | % | Canis lupus familiaris | |||
16. | ALA4078272 | 3-(S) | t1/2 | = | 7.5 | hr | ALA4012163 | hr | Canis lupus familiaris | |||
17. | ALA4078272 | 3-(S) | Vd | = | 0.7 | l | ALA4012161 | l | Canis lupus familiaris | |||
18. | ALA4078272 | 3-(S) | CL | = | 1.4 | ml/min.kg | ALA4012160 | mL.min-1.kg-1 | Canis lupus familiaris | |||
19. | ALA4078272 | 3-(S) | solubility | = | 34 | uM | ALA4012159 | nM | ||||
20. | ALA4078272 | 3-(S) | solubility | = | 40 | uM | ALA4012158 | nM |