| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4080789 | 6d | Activity | 0 | ALA4030890 | Active | Rattus norvegicus | |||||
| 2. | ALA4080789 | 6d | K | = | 2.3 | 10'-3/s | ALA4030899 | 10'-3/s | Homo sapiens | |||
| 3. | ALA4080789 | 6d | K | = | 8.1 | 10'3/M/s | ALA4030898 | 10'3/M/s | Homo sapiens | |||
| 4. | ALA4080789 | 6d | INH | 0 | ALA4030897 | Active | % | Mus musculus | ||||
| 5. | ALA4080789 | 6d | INH | 0 | ALA4030896 | Active | % | Mus musculus | ||||
| 6. | ALA4080789 | 6d | Activity | 0 | ALA4030895 | Active | ||||||
| 7. | ALA4080789 | 6d | Activity | 0 | ALA4030894 | Not Active | Homo sapiens | |||||
| 8. | ALA4080789 | 6d | Activity | 0 | ALA4030893 | Active | Homo sapiens | |||||
| 9. | ALA4080789 | 6d | Activity | 0 | ALA4030892 | Not Active | Rattus norvegicus | |||||
| 10. | ALA4080789 | 6d | Activity | 0 | ALA4030891 | Active | Rattus norvegicus | |||||
| 11. | ALA4080789 | 6d | t1/2 | = | 39.8 | min | ALA4030889 | hr | Rattus norvegicus | |||
| 12. | ALA4080789 | 6d | t1/2 | = | 85.6 | min | ALA4030888 | hr | Rattus norvegicus | |||
| 13. | ALA4080789 | 6d | t1/2 | = | 126.5 | min | ALA4030887 | hr | Rattus norvegicus | |||
| 14. | ALA4080789 | 6d | F | = | 16.8 | % | ALA4030886 | % | Rattus norvegicus | |||
| 15. | ALA4080789 | 6d | AUC | = | 314 | ng.hr/ml | ALA4030885 | ng.hr.mL-1 | Rattus norvegicus | |||
| 16. | ALA4080789 | 6d | t1/2 | = | 2.86 | hr | ALA4030884 | hr | Rattus norvegicus | |||
| 17. | ALA4080789 | 6d | Cmax | = | 42.2 | ng/ml | ALA4030883 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 18. | ALA4080789 | 6d | Tmax | = | 3.83 | hr | ALA4030882 | hr | Rattus norvegicus | |||
| 19. | ALA4080789 | 6d | CL | = | 2.48 | L/hr/kg | ALA4030856 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 20. | ALA4080789 | 6d | AUC | = | 408 | ng.hr/ml | ALA4030857 | ng.hr.mL-1 | Rattus norvegicus |
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