# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4081385 | 28f | FC | = | 80 | ALA4022804 | Mus musculus | |||||
2. | ALA4081385 | 28f | FC | > | 100 | ALA4022803 | Mus musculus | |||||
3. | ALA4081385 | 28f | F | = | 33 | % | ALA4022802 | % | Mus musculus | |||
4. | ALA4081385 | 28f | fCmax | = | 232 | nM | ALA4022801 | nM | Mus musculus | |||
5. | ALA4081385 | 28f | t1/2 | = | 2.8 | hr | ALA4022800 | hr | Mus musculus | |||
6. | ALA4081385 | 28f | fAUC | = | 1520 | nM.hr | ALA4022799 | uM.hr | Mus musculus | |||
7. | ALA4081385 | 28f | Vduss | = | 9 | L/Kg | ALA4022798 | L.kg-1 | Mus musculus | |||
8. | ALA4081385 | 28f | CL free | = | 44 | ml/min.kg | ALA4022797 | mL.min-1.kg-1 | Mus musculus | |||
9. | ALA4081385 | 28f | Fu | = | 0.05 | ALA4022785 | Mus musculus | |||||
10. | ALA4081385 | 28f | Cp | = | 9.1 | uM | ALA4022784 | uM | Mus musculus | |||
11. | ALA4081385 | 28f | permeability | = | 0.18 | % | ALA4022780 | % | ||||
12. | ALA4081385 | 28f | EC50 | = | 7.9 | nM | ALA4022774 | 8.10 | nM | Homo sapiens | ||
13. | ALA4081385 | 28f | IC50 | = | 7.8 | nM | ALA4022773 | 8.11 | nM | Homo sapiens |