# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4082531 | 2 | IC50 | = | 0.84 | uM | ALA4008879 | 6.08 | nM | Homo sapiens | ||
2. | ALA4082531 | 2 | IC50 | = | 21.3 | uM | ALA4008878 | 4.67 | nM | Homo sapiens | ||
3. | ALA4082531 | 2 | IC50 | = | 0.8 | uM | ALA4008877 | 6.10 | nM | Homo sapiens | ||
4. | ALA4082531 | 2 | IC50 | = | 2.1 | uM | ALA4008872 | 5.68 | nM | Homo sapiens | ||
5. | ALA4082531 | 2 | IC50 | = | 47 | uM | ALA4008865 | 4.33 | nM | Homo sapiens | ||
6. | ALA4082531 | 2 | CL/F | = | 2.32 | g/min | ALA3998703 | g/min | ||||
7. | ALA4082531 | 2 | Vz/F | = | 1720 | g | ALA3998702 | g | ||||
8. | ALA4082531 | 2 | AUClast | = | 885986 | min.ng/g | ALA3998701 | min.ng/g | ||||
9. | ALA4082531 | 2 | Tmax | = | 30 | min | ALA3998700 | hr | ||||
10. | ALA4082531 | 2 | Cmax | = | 17426 | ng/g | ALA3998699 | ng/g | ||||
11. | ALA4082531 | 2 | beta t1/2 | = | 514 | min | ALA3998698 | hr | ||||
12. | ALA4082531 | 2 | CL/F | = | 8.13 | g/min | ALA3998697 | g/min | Mus musculus | |||
13. | ALA4082531 | 2 | Vz/F | = | 1174 | g | ALA3998696 | g | Mus musculus | |||
14. | ALA4082531 | 2 | AUClast | = | 245088 | min.ng/g | ALA3998695 | min.ng/g | Mus musculus | |||
15. | ALA4082531 | 2 | Tmax | = | 10 | min | ALA3998694 | hr | Mus musculus | |||
16. | ALA4082531 | 2 | Cmax | = | 5707 | ng/g | ALA3998693 | ng/g | Mus musculus | |||
17. | ALA4082531 | 2 | beta t1/2 | = | 100 | min | ALA3998692 | hr | Mus musculus | |||
18. | ALA4082531 | 2 | CL/F | = | 1.39 | ml/min | ALA3998691 | ml/min | Mus musculus | |||
19. | ALA4082531 | 2 | Vz/F | = | 679 | ml | ALA3998690 | ml | Mus musculus | |||
20. | ALA4082531 | 2 | AUClast | = | 1494106 | min.ng/ml | ALA3998689 | ng.hr.mL-1 | Mus musculus |