| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4083687 | 3 | Emax | = | 68 | % | ALA4251999 | % | Homo sapiens | |||
| 2. | ALA4083687 | 3 | Emax | = | 108 | % | ALA4252017 | % | Homo sapiens | |||
| 3. | ALA4083687 | 3 | Kd | = | 0.07 | uM | ALA4252018 | 7.16 | nM | Homo sapiens | ||
| 4. | ALA4083687 | 3 | EC50 | = | 0.3 | uM | ALA4252017 | 6.52 | nM | Homo sapiens | ||
| 5. | ALA4083687 | 3 | CLH | = | 1420 | uL/min.mg | ALA4252004 | mL.min-1.g-1 | ||||
| 6. | ALA4083687 | 3 | solubility | < | 1 | uM | ALA4252003 | nM | ||||
| 7. | ALA4083687 | 3 | Ratio | = | 0.8 | ALA4252002 | ||||||
| 8. | ALA4083687 | 3 | Ratio | = | 0.8 | ALA4252001 | ||||||
| 9. | ALA4083687 | 3 | Papp | = | 44 | ucm/s | ALA4252000 | ucm/s | ||||
| 10. | ALA4083687 | 3 | EC50 | = | 0.37 | uM | ALA4251999 | 6.43 | nM | Homo sapiens | ||
| 11. | ALA4083687 | 3 | fCmax | = | 0.07 | uM | ALA3993216 | uM | Mus musculus | |||
| 12. | ALA4083687 | 3 | Drug metabolism | 0 | ALA3993214 | Metabolite_Detected | Mus musculus | |||||
| 13. | ALA4083687 | 3 | Drug metabolism | 0 | ALA3993213 | Metabolite_Detected | Mus musculus | |||||
| 14. | ALA4083687 | 3 | Drug metabolism | 0 | ALA3993212 | Metabolite_Detected | Mus musculus | |||||
| 15. | ALA4083687 | 3 | Ratio | = | 0.8 | ALA3993211 | ||||||
| 16. | ALA4083687 | 3 | Ratio | = | 0.8 | ALA3993210 | ||||||
| 17. | ALA4083687 | 3 | Papp | = | 46 | ucm/s | ALA3993209 | ucm/s | ||||
| 18. | ALA4083687 | 3 | CLH | = | 1420 | microL/min/mg | ALA3993208 | mL.min-1.g-1 | Mus musculus | |||
| 19. | ALA4083687 | 3 | MEC | = | 0.78 | uM | ALA3993207 | uM | Homo sapiens |
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