| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4084135 | 56 | K(p,uu,brain) | = | 0.42 | ALA4037534 | ||||||
| 2. | ALA4084135 | 56 | AUC/dose | = | 13.4 | ng.hr/g/mg/kg | ALA4037532 | ng.hr/g/mg/kg | Rattus norvegicus | |||
| 3. | ALA4084135 | 56 | Fu | = | 3.3 | % | ALA4037529 | Rattus norvegicus | ||||
| 4. | ALA4084135 | 56 | pIC50 | = | 6.5 | ALA4037528 | 6.50 | nM | Homo sapiens | |||
| 5. | ALA4084135 | 56 | Kp | = | 0.21 | ALA4037533 | ||||||
| 6. | ALA4084135 | 56 | AUC/dose | = | 63.8 | ng.hr/ml/mg/kg | ALA4037531 | ng.hr/ml/mg/kg | Rattus norvegicus | |||
| 7. | ALA4084135 | 56 | Fu | = | 1.6 | % | ALA4037530 | Rattus norvegicus | ||||
| 8. | ALA4084135 | 56 | pIC50 | = | 8.8 | ALA4037524 | 8.80 | nM | Homo sapiens | |||
| 9. | ALA4084135 | 56 | solubility | = | 25.2 | ug ml-1 | ALA4037525 | ug.mL-1 | ||||
| 10. | ALA4084135 | 56 | Ratio | = | 2.2 | ALA4037526 | Canis lupus familiaris | |||||
| 11. | ALA4084135 | 56 | permeability | = | 331 | nm/s | ALA4037527 | nm/s | Canis lupus familiaris |
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