| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4084621 | 1c; BMS-933043 | Activity | 0 | ALA4004708 | Not Active | Homo sapiens | |||||
| 2. | ALA4084621 | 1c; BMS-933043 | Ratio EC50 | > | 100 | ALA4004778 | ||||||
| 3. | ALA4084621 | 1c; BMS-933043 | Ratio EC50 | > | 100 | ALA4004777 | ||||||
| 4. | ALA4084621 | 1c; BMS-933043 | Ratio EC50 | > | 100 | ALA4004776 | ||||||
| 5. | ALA4084621 | 1c; BMS-933043 | Drug metabolism | 0 | ALA4004774 | Metabolite_Detected | ||||||
| 6. | ALA4084621 | 1c; BMS-933043 | Ratio | > | 600 | ALA4004773 | ||||||
| 7. | ALA4084621 | 1c; BMS-933043 | Fu | = | 84 | % | ALA4004733 | Mus musculus | ||||
| 8. | ALA4084621 | 1c; BMS-933043 | MED | = | 0.1 | mg kg-1 | ALA4004766 | mg kg-1 | Mus musculus | |||
| 9. | ALA4084621 | 1c; BMS-933043 | Stability | = | 93 | % | ALA4004769 | % | Mus musculus | |||
| 10. | ALA4084621 | 1c; BMS-933043 | F | = | 70 | % | ALA4004764 | % | Macaca fascicularis | |||
| 11. | ALA4084621 | 1c; BMS-933043 | AUC | = | 11 | uM.hr | ALA4004763 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Macaca fascicularis | ||
| 12. | ALA4084621 | 1c; BMS-933043 | Cmax | = | 1.3 | uM | ALA4004762 | nM | Macaca fascicularis | |||
| 13. | ALA4084621 | 1c; BMS-933043 | AUC | = | 3 | uM.hr | ALA4004761 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Macaca fascicularis | ||
| 14. | ALA4084621 | 1c; BMS-933043 | t1/2 | = | 4.4 | hr | ALA4004760 | hr | Macaca fascicularis | |||
| 15. | ALA4084621 | 1c; BMS-933043 | CL | = | 17 | ml/min.kg | ALA4004759 | mL.min-1.kg-1 | Macaca fascicularis | |||
| 16. | ALA4084621 | 1c; BMS-933043 | Vdss | = | 5.7 | L/Kg | ALA4004758 | L.kg-1 | Macaca fascicularis | |||
| 17. | ALA4084621 | 1c; BMS-933043 | F | = | 100 | % | ALA4004757 | % | Canis lupus familiaris | |||
| 18. | ALA4084621 | 1c; BMS-933043 | AUC | = | 19 | uM.hr | ALA4004756 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Canis lupus familiaris | ||
| 19. | ALA4084621 | 1c; BMS-933043 | Cmax | = | 3.2 | uM | ALA4004755 | nM | Canis lupus familiaris | |||
| 20. | ALA4084621 | 1c; BMS-933043 | AUC | = | 3.4 | uM.hr | ALA4004754 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Canis lupus familiaris |
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