| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4084855 | 29 | IC50 | = | 25 | uM | ALA4057843 | 4.60 | nM | Homo sapiens | ||
| 2. | ALA4084855 | 29 | IC50 | > | 25 | uM | ALA4057842 | nM | Homo sapiens | |||
| 3. | ALA4084855 | 29 | IC50 | = | 18 | uM | ALA4057841 | 4.75 | nM | Homo sapiens | ||
| 4. | ALA4084855 | 29 | CLH | = | 0.09 | ml/min/mg | ALA4057840 | mL.min-1.g-1 | Homo sapiens | |||
| 5. | ALA4084855 | 29 | IC50 | = | 0.1 | nM | ALA4057839 | 10.00 | nM | Homo sapiens | ||
| 6. | ALA4084855 | 29 | INH | = | 60 | % | ALA4057837 | % | Mus musculus | |||
| 7. | ALA4084855 | 29 | Kp | = | 2.1 | ALA4057849 | ||||||
| 8. | ALA4084855 | 29 | Kp | = | 2.1 | ALA4057850 | ||||||
| 9. | ALA4084855 | 29 | Activity | 0 | ALA4057851 | Non-Toxic | Mus musculus | |||||
| 10. | ALA4084855 | 29 | permeability | = | 610 | 10'-7 cm/s | ALA4057844 | 10'-7 cm/s | ||||
| 11. | ALA4084855 | 29 | Cmax | = | 248 | ng/ml | ALA4057845 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Mus musculus | ||
| 12. | ALA4084855 | 29 | Cmax | = | 528 | ng/ml | ALA4057846 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Mus musculus | ||
| 13. | ALA4084855 | 29 | AUC | = | 770 | ng.hr/ml | ALA4057847 | ng.hr.mL-1 | Mus musculus | |||
| 14. | ALA4084855 | 29 | AUC | = | 1614 | ng.hr/ml | ALA4057848 | ng.hr.mL-1 | Mus musculus |
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