# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4086264 | 6b | Ratio IC50 | > | 1000 | ALA4021465 | ||||||
2. | ALA4086264 | 6b | Ratio IC50 | > | 1000 | ALA4021464 | ||||||
3. | ALA4086264 | 6b | Ratio IC50 | > | 1000 | ALA4021463 | ||||||
4. | ALA4086264 | 6b | Ratio IC50 | > | 1000 | ALA4021462 | ||||||
5. | ALA4086264 | 6b | Ratio IC50 | = | 11.6 | ALA4021461 | ||||||
6. | ALA4086264 | 6b | Ratio IC50 | = | 2.8 | ALA4021460 | ||||||
7. | ALA4086264 | 6b | Ratio IC50 | = | 8.6 | ALA4021459 | ||||||
8. | ALA4086264 | 6b | Ratio IC50 | = | 5.6 | ALA4021458 | ||||||
9. | ALA4086264 | 6b | AUC | = | 2.86 | microg.hr/mL | ALA4021457 | ng.hr.mL-1 | Rattus norvegicus | |||
10. | ALA4086264 | 6b | AUC | = | 2.36 | microg.hr/mL | ALA4021456 | ng.hr.mL-1 | Rattus norvegicus | |||
11. | ALA4086264 | 6b | Cmax | = | 0.55 | ug ml-1 | ALA4021455 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
12. | ALA4086264 | 6b | Tmax | = | 1.67 | hr | ALA4021454 | hr | Rattus norvegicus | |||
13. | ALA4086264 | 6b | permeability | 0 | ALA4021453 | Permeable | ||||||
14. | ALA4086264 | 6b | Stability | 0 | ALA4021452 | Stable | % | Canis lupus familiaris | ||||
15. | ALA4086264 | 6b | Stability | 0 | ALA4021451 | Stable | % | Rattus norvegicus | ||||
16. | ALA4086264 | 6b | Stability | 0 | ALA4021450 | Stable | % | Mus musculus | ||||
17. | ALA4086264 | 6b | Stability | 0 | ALA4021427 | Stable | % | Homo sapiens | ||||
18. | ALA4086264 | 6b | INH | 0 | ALA4021449 | Not Active | % | Homo sapiens | ||||
19. | ALA4086264 | 6b | INH | 0 | ALA4021448 | Not Active | % | Homo sapiens | ||||
20. | ALA4086264 | 6b | INH | 0 | ALA4021426 | Not Active | % | Homo sapiens |