| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4086957 | 42 | Ratio | = | 2.4 | ALA4037616 | ||||||
| 2. | ALA4086957 | 42 | K(p,uu,brain) | 0 | ALA4037534 | Not Determined | ||||||
| 3. | ALA4086957 | 42 | AUC/dose | = | 243 | ng.hr/g/mg/kg | ALA4037532 | ng.hr/g/mg/kg | Rattus norvegicus | |||
| 4. | ALA4086957 | 42 | Fu | = | 0.65 | % | ALA4037530 | Rattus norvegicus | ||||
| 5. | ALA4086957 | 42 | pIC50 | = | 6.2 | ALA4037528 | 6.20 | nM | Homo sapiens | |||
| 6. | ALA4086957 | 42 | Kp | = | 0.06 | ALA4037533 | ||||||
| 7. | ALA4086957 | 42 | Fu | = | 5.1 | % | ALA4037529 | Rattus norvegicus | ||||
| 8. | ALA4086957 | 42 | AUC/dose | = | 4331 | ng.hr/ml/mg/kg | ALA4037531 | ng.hr/ml/mg/kg | Rattus norvegicus | |||
| 9. | ALA4086957 | 42 | pIC50 | = | 9.4 | ALA4037524 | 9.40 | nM | Homo sapiens | |||
| 10. | ALA4086957 | 42 | solubility | = | 50.8 | ug ml-1 | ALA4037525 | ug.mL-1 | ||||
| 11. | ALA4086957 | 42 | permeability | = | 348 | nm/s | ALA4037527 | nm/s | Canis lupus familiaris |
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