# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4089543 | [3H]33 | Bmax | = | 1800 | disintegrations/minute | ALA4051394 | disintegrations/minute | Homo sapiens | |||
2. | ALA4089543 | [3H]33 | Kd(app) | = | 0.22 | nM | ALA4051395 | 9.66 | nM | Homo sapiens | ||
3. | ALA4089543 | [3H]33 | pIC50 | = | 4.73 | ALA4051424 | 4.73 | nM | Homo sapiens | |||
4. | ALA4089543 | [3H]33 | pIC50 | = | 4.98 | ALA4051423 | 4.98 | nM | Homo sapiens | |||
5. | ALA4089543 | [3H]33 | pIC50 | = | 5.18 | ALA4051422 | 5.18 | nM | Homo sapiens | |||
6. | ALA4089543 | [3H]33 | pIC50 | = | 5.57 | ALA4051421 | 5.57 | nM | Homo sapiens | |||
7. | ALA4089543 | [3H]33 | Activity | < | 15 | % | ALA4051414 | % | Homo sapiens | |||
8. | ALA4089543 | [3H]33 | Activity | > | 60 | % | ALA4051413 | % | Homo sapiens | |||
9. | ALA4089543 | [3H]33 | Stability | 0 | ALA4051411 | Unstable | % | |||||
10. | ALA4089543 | [3H]33 | Kd | = | 0.31 | nM | ALA4051407 | 9.51 | nM | Homo sapiens | ||
11. | ALA4089543 | [3H]33 | Kd | = | 0.2 | nM | ALA4051405 | 9.70 | nM | Homo sapiens | ||
12. | ALA4089543 | [3H]33 | Ki | = | 0.41 | nM | ALA4051384 | 9.39 | nM | Homo sapiens | ||
13. | ALA4089543 | [3H]33 | Kd | = | 0.91 | nM | ALA4051393 | 9.04 | nM | Homo sapiens | ||
14. | ALA4089543 | [3H]33 | Bmax | = | 1200 | disintegrations/minute | ALA4051393 | disintegrations/minute | Homo sapiens | |||
15. | ALA4089543 | [3H]33 | Kd(app) | = | 0.31 | nM | ALA4051394 | 9.51 | nM | Homo sapiens | ||
16. | ALA4089543 | [3H]33 | Bmax | = | 620 | disintegrations/minute | ALA4051395 | disintegrations/minute | Homo sapiens | |||
17. | ALA4089543 | [3H]33 | Kd | = | 0.67 | nM | ALA4051396 | 9.17 | nM | Homo sapiens | ||
18. | ALA4089543 | [3H]33 | K | = | 0.056 | /min/nM | ALA4051402 | /min/nM | Homo sapiens | |||
19. | ALA4089543 | [3H]33 | K | = | 0.011 | /min | ALA4051403 | /min | Homo sapiens | |||
20. | ALA4089543 | [3H]33 | t1/2 | = | 66 | min | ALA4051404 | hr | Homo sapiens |