# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4092369 | 31; GPA | IC50 | = | 4.9 | nM | ALA3992745 | 8.31 | nM | Homo sapiens | ||
2. | ALA4092369 | 31; GPA | Activity | 0 | ALA5035158 | Toxic | ||||||
3. | ALA4092369 | 31; GPA | Drug metabolism | = | 14.87 | ng/ml | ALA5035157 | ng/ml | ||||
4. | ALA4092369 | 31; GPA | Drug metabolism | 0 | ALA5035156 | Metabolite_Detected | ||||||
5. | ALA4092369 | 31; GPA | Drug uptake | = | 35.4 | ng/ml | ALA5035155 | ng/ml | ||||
6. | ALA4092369 | 31; GPA | Kd | = | 3.492 | M | ALA5035154 | nM | Homo sapiens | |||
7. | ALA4092369 | 31; GPA | Cmax | = | 18.45 | ng/ml | ALA5035153 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
8. | ALA4092369 | 31; GPA | Activity | = | 38 | % | ALA5035152 | % | ||||
9. | ALA4092369 | 31; GPA | Activity | = | 51 | % | ALA5035151 | % | ||||
10. | ALA4092369 | 31; GPA | Activity | 0 | ALA5035150 | Active | ||||||
11. | ALA4092369 | 31; GPA | Activity | 0 | ALA5035149 | Not Active | ||||||
12. | ALA4092369 | 31; GPA | FC | = | 2.2 | ALA5035148 | ||||||
13. | ALA4092369 | 31; GPA | FC | = | 2.5 | ALA5035147 | ||||||
14. | ALA4092369 | 31; GPA | FC | = | 3.6 | ALA5035146 | ||||||
15. | ALA4092369 | 31; GPA | FC | = | 3.6 | ALA5035145 | ||||||
16. | ALA4092369 | 31; GPA | Activity | = | 61 | % | ALA5035144 | % | ||||
17. | ALA4092369 | 31; GPA | Activity | 0 | ALA5035140 | Non-Toxic | Homo sapiens | |||||
18. | ALA4092369 | 31; GPA | Activity | 0 | ALA5035139 | Not Active | ||||||
19. | ALA4092369 | 31; GPA | Activity | 0 | ALA5035138 | Not Active | ||||||
20. | ALA4092369 | 31; GPA | Activity | = | 86 | % | ALA5035137 | % |