| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4092752 | 4 | F | = | 19 | % | ALA4022545 | % | Macaca mulatta | |||
| 2. | ALA4092752 | 4 | AUC | = | 10 | uM.hr | ALA4022543 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Macaca mulatta | ||
| 3. | ALA4092752 | 4 | F | = | 98 | % | ALA4022542 | % | Canis lupus familiaris | |||
| 4. | ALA4092752 | 4 | AUC | = | 52 | uM.hr | ALA4022540 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Canis lupus familiaris | ||
| 5. | ALA4092752 | 4 | F | = | 58 | % | ALA4022539 | % | Rattus norvegicus | |||
| 6. | ALA4092752 | 4 | AUC | = | 11 | uM.hr | ALA4022538 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 7. | ALA4092752 | 4 | CL | = | 7 | ml/min.kg | ALA4022537 | mL.min-1.kg-1 | Macaca mulatta | |||
| 8. | ALA4092752 | 4 | CL | = | 23 | ml/min.kg | ALA4022536 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 9. | ALA4092752 | 4 | CL | = | 3 | ml/min.kg | ALA4022535 | mL.min-1.kg-1 | Canis lupus familiaris | |||
| 10. | ALA4092752 | 4 | permeability | = | 15 | nm/s | ALA4022534 | nm/s | ||||
| 11. | ALA4092752 | 4 | AUC | = | 13 | uM.hr | ALA4022533 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 12. | ALA4092752 | 4 | IC50 | = | 0.27 | uM | ALA4022532 | 6.57 | nM | Homo sapiens | ||
| 13. | ALA4092752 | 4 | Ki | = | 0.7 | nM | ALA4022531 | 9.15 | nM | Homo sapiens | ||
| 14. | ALA4092752 | 4 | IC50 | = | 144 | nM | ALA4022530 | 6.84 | nM | Homo sapiens | ||
| 15. | ALA4092752 | 4 | IC50 | = | 239 | nM | ALA4022529 | 6.62 | nM | Homo sapiens | ||
| 16. | ALA4092752 | 4 | IC50 | = | 684 | nM | ALA4022528 | 6.17 | nM | Homo sapiens | ||
| 17. | ALA4092752 | 4 | IC50 | = | 1760 | nM | ALA4022527 | 5.75 | nM | Homo sapiens | ||
| 18. | ALA4092752 | 4 | IC50 | > | 40000 | nM | ALA4022526 | nM | Homo sapiens | |||
| 19. | ALA4092752 | 4 | IC50 | = | 5500 | nM | ALA4022525 | 5.26 | nM | Homo sapiens | ||
| 20. | ALA4092752 | 4 | IC50 | = | 533 | nM | ALA4022524 | 6.27 | nM | Homo sapiens |
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