# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4093031 | 37; BMS-929075 | Vdss | = | 0.7 | L/Kg | ALA4015605 | L.kg-1 | Rattus norvegicus | |||
2. | ALA4093031 | 37; BMS-929075 | Cmax | = | 7.5 | uM | ALA4015606 | nM | Rattus norvegicus | |||
3. | ALA4093031 | 37; BMS-929075 | Tmax | = | 4 | hr | ALA4015607 | hr | Rattus norvegicus | |||
4. | ALA4093031 | 37; BMS-929075 | AUC | = | 54.5 | uM.hr | ALA4015608 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
5. | ALA4093031 | 37; BMS-929075 | F | > | 100 | % | ALA4015642 | % | Rattus norvegicus | |||
6. | ALA4093031 | 37; BMS-929075 | Activity | 0 | ALA4015609 | Active | Hepacivirus hominis | |||||
7. | ALA4093031 | 37; BMS-929075 | Drug uptake | = | 1.12 | uM | ALA4015610 | uM | Rattus norvegicus | |||
8. | ALA4093031 | 37; BMS-929075 | Ratio | = | 10 | ALA4015598 | ||||||
9. | ALA4093031 | 37; BMS-929075 | Ratio | = | 10 | ALA4015599 | ||||||
10. | ALA4093031 | 37; BMS-929075 | Activity | 0 | ALA4015600 | Non-Toxic | Canis lupus familiaris | |||||
11. | ALA4093031 | 37; BMS-929075 | Activity | 0 | ALA4015636 | Non-Toxic | Rattus norvegicus | |||||
12. | ALA4093031 | 37; BMS-929075 | AUC | = | 140.2 | uM.hr | ALA4015635 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
13. | ALA4093031 | 37; BMS-929075 | Tmax | = | 4 | hr | ALA4015634 | hr | Rattus norvegicus | |||
14. | ALA4093031 | 37; BMS-929075 | Cmax | = | 14.7 | uM | ALA4015633 | nM | Rattus norvegicus | |||
15. | ALA4093031 | 37; BMS-929075 | solubility | < | 1 | ug ml-1 | ALA4015632 | ug.mL-1 | ||||
16. | ALA4093031 | 37; BMS-929075 | Peff | > | 100 | nm/s | ALA4015631 | nm/s | ||||
17. | ALA4093031 | 37; BMS-929075 | CC50 | > | 50 | uM | ALA4015622 | nM | Homo sapiens | |||
18. | ALA4093031 | 37; BMS-929075 | CC50 | > | 12.5 | uM | ALA4015627 | nM | Homo sapiens | |||
19. | ALA4093031 | 37; BMS-929075 | logD | = | 3.3 | ALA4015626 | ||||||
20. | ALA4093031 | 37; BMS-929075 | Activity | 0 | ALA4015623 | Active | Hepacivirus hominis |