# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4095192 | 5b | MTC | = | 5.4 | mg kg-1 | ALA4009211 | mg kg-1 | Mus musculus | |||
2. | ALA4095192 | 5b | ED50 | = | 2.2 | mg kg-1 | ALA4009210 | mg.kg-1 | Mus musculus | |||
3. | ALA4095192 | 5b | INH | = | 66 | % | ALA4009190 | % | Mus musculus | |||
4. | ALA4095192 | 5b | INH | = | 41 | % | ALA4009189 | % | Mus musculus | |||
5. | ALA4095192 | 5b | INH | = | 25 | % | ALA4009188 | % | Mus musculus | |||
6. | ALA4095192 | 5b | INH | = | 23 | % | ALA4009187 | % | Mus musculus | |||
7. | ALA4095192 | 5b | Activity | = | 113 | % | ALA4009153 | % | Homo sapiens | |||
8. | ALA4095192 | 5b | EC50 | = | 0.9 | nM | ALA4009152 | 9.05 | nM | Homo sapiens | ||
9. | ALA4095192 | 5b | INH | = | 21 | % | ALA4009150 | % | ||||
10. | ALA4095192 | 5b | INH | = | 12 | % | ALA4009148 | % | ||||
11. | ALA4095192 | 5b | INH | = | 0 | % | ALA4009146 | % | Cavia porcellus | |||
12. | ALA4095192 | 5b | Ki | = | 101 | nM | ALA4009144 | 7.00 | nM | |||
13. | ALA4095192 | 5b | Ki | = | 184 | nM | ALA4009142 | 6.74 | nM | Cavia porcellus | ||
14. | ALA4095192 | 5b | Ki | = | 0.45 | nM | ALA4009141 | 9.35 | nM | Cavia porcellus |