| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4095883 | 7 | Selectivity ratio | > | 1000 | ALA4040346 | ||||||
| 2. | ALA4095883 | 7 | Drug uptake | 0 | ALA4040345 | Active | ||||||
| 3. | ALA4095883 | 7 | Drug uptake | 0 | ALA4040344 | Active | ||||||
| 4. | ALA4095883 | 7 | Drug uptake | 0 | ALA4040343 | Active | ||||||
| 5. | ALA4095883 | 7 | Activity | 0 | ALA4040342 | Toxic | Rattus norvegicus | |||||
| 6. | ALA4095883 | 7 | Activity | 0 | ALA4040341 | Toxic | Rattus norvegicus | |||||
| 7. | ALA4095883 | 7 | Selectivity Index | > | 4000 | ALA4040340 | Homo sapiens | |||||
| 8. | ALA4095883 | 7 | Activity | = | 54 | % | ALA4040339 | % | Homo sapiens | |||
| 9. | ALA4095883 | 7 | Ratio | = | 2 | ALA4040338 | ||||||
| 10. | ALA4095883 | 7 | Efficacy | = | 46 | % | ALA4040337 | % | Homo sapiens | |||
| 11. | ALA4095883 | 7 | EC50 | = | 1205.8 | nM | ALA4040336 | 5.92 | nM | Homo sapiens | ||
| 12. | ALA4095883 | 7 | Efficacy | = | 91 | % | ALA4040302 | % | Homo sapiens | |||
| 13. | ALA4095883 | 7 | EC50 | = | 0.34 | nM | ALA4040335 | 9.47 | nM | Homo sapiens | ||
| 14. | ALA4095883 | 7 | Activity | 0 | ALA4040301 | Active | Rattus norvegicus | |||||
| 15. | ALA4095883 | 7 | Activity | 0 | ALA4040328 | Non-Toxic | Rattus norvegicus | |||||
| 16. | ALA4095883 | 7 | Activity | 0 | ALA4040329 | Non-Toxic | Rattus norvegicus | |||||
| 17. | ALA4095883 | 7 | Activity | 0 | ALA4040333 | Toxic | Rattus norvegicus | |||||
| 18. | ALA4095883 | 7 | IC50 | = | 3.2 | nM | ALA4040321 | 8.49 | nM | Homo sapiens | ||
| 19. | ALA4095883 | 7 | solubility | = | 146 | uM | ALA4040304 | nM | ||||
| 20. | ALA4095883 | 7 | CLH | = | 40 | microL/min/mg | ALA4040305 | mL.min-1.g-1 | Homo sapiens |
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