# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | GNE-781 | 19 | INH | 0 | ALA4058652 | Dose-dependent effect | % | Homo sapiens | ||||
2. | GNE-781 | 19 | Drug uptake | 0 | ALA4058667 | Active | ||||||
3. | GNE-781 | 19 | Drug uptake | 0 | ALA4058666 | Active | Mus musculus | |||||
4. | GNE-781 | 19 | Activity | = | 150 | % | ALA4058665 | % | Mus musculus | |||
5. | GNE-781 | 19 | INH | 0 | ALA4058664 | Active | % | Mus musculus | ||||
6. | GNE-781 | 19 | IC50 | > | 10 | uM | ALA4058663 | nM | Homo sapiens | |||
7. | GNE-781 | 19 | IC50 | > | 10 | uM | ALA4058662 | nM | Homo sapiens | |||
8. | GNE-781 | 19 | Ratio IC50 | = | 5425 | ALA4058602 | ||||||
9. | GNE-781 | 19 | IC50 | = | 6.2 | nM | ALA4058603 | 8.21 | nM | Homo sapiens | ||
10. | GNE-781 | 19 | IC50 | = | 0.94 | nM | ALA4058600 | 9.03 | nM | Homo sapiens | ||
11. | GNE-781 | 19 | EC50 | = | 6.6 | nM | ALA4058604 | 8.18 | nM | Homo sapiens | ||
12. | GNE-781 | 19 | IC50 | = | 1.2 | nM | ALA4058605 | 8.92 | nM | Homo sapiens | ||
13. | GNE-781 | 19 | IC50 | > | 18000 | nM | ALA4058606 | nM | Homo sapiens | |||
14. | GNE-781 | 19 | IC50 | > | 20000 | nM | ALA4058607 | nM | Homo sapiens | |||
15. | GNE-781 | 19 | IC50 | = | 12000 | nM | ALA4058608 | 4.92 | nM | Homo sapiens | ||
16. | GNE-781 | 19 | IC50 | > | 20000 | nM | ALA4058609 | nM | Homo sapiens | |||
17. | GNE-781 | 19 | IC50 | > | 20000 | nM | ALA4058610 | nM | Homo sapiens | |||
18. | GNE-781 | 19 | IC50 | = | 4600 | nM | ALA4058611 | 5.34 | nM | Homo sapiens | ||
19. | GNE-781 | 19 | IC50 | > | 20000 | nM | ALA4058612 | nM | Homo sapiens | |||
20. | GNE-781 | 19 | IC50 | > | 20000 | nM | ALA4058613 | nM | Homo sapiens |