| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4097298 | 25 | EC50 | = | 3.6 | uM | ALA4016946 | 5.44 | nM | Rattus norvegicus | ||
| 2. | ALA4097298 | 25 | ED50 | = | 40 | mg kg-1 | ALA4016945 | mg.kg-1 | Rattus norvegicus | |||
| 3. | ALA4097298 | 25 | Time | <= | 7 | hr | ALA4016943 | hr | Rattus norvegicus | |||
| 4. | ALA4097298 | 25 | F | = | 50 | % | ALA4016942 | % | Rattus norvegicus | |||
| 5. | ALA4097298 | 25 | AUC | = | 10220 | ng.hr/ml | ALA4016941 | ng.hr.mL-1 | Rattus norvegicus | |||
| 6. | ALA4097298 | 25 | t1/2 | = | 3.3 | hr | ALA4016940 | hr | Rattus norvegicus | |||
| 7. | ALA4097298 | 25 | IC50 | = | 27 | nM | ALA4016909 | 7.57 | nM | Homo sapiens | ||
| 8. | ALA4097298 | 25 | IC50 | = | 2 | nM | ALA4016908 | 8.70 | nM | Homo sapiens | ||
| 9. | ALA4097298 | 25 | Ratio IC50 | = | 14 | ALA4016910 | ||||||
| 10. | ALA4097298 | 25 | IC50 | = | 1.8 | uM | ALA4016911 | 5.75 | nM | Rattus norvegicus | ||
| 11. | ALA4097298 | 25 | Ratio IC50 | = | 1000 | ALA4016912 | ||||||
| 12. | ALA4097298 | 25 | t1/2 | = | 125 | min | ALA4016913 | hr | Homo sapiens | |||
| 13. | ALA4097298 | 25 | t1/2 | = | 23 | min | ALA4016914 | hr | Rattus norvegicus | |||
| 14. | ALA4097298 | 25 | INH | <= | 9 | % | ALA4016915 | % | Homo sapiens | |||
| 15. | ALA4097298 | 25 | INH | <= | 9 | % | ALA4016916 | % | Homo sapiens | |||
| 16. | ALA4097298 | 25 | INH | = | 23 | % | ALA4016917 | % | Homo sapiens | |||
| 17. | ALA4097298 | 25 | INH | = | 19 | % | ALA4016918 | % | Homo sapiens | |||
| 18. | ALA4097298 | 25 | INH | = | 17 | % | ALA4016919 | % | Homo sapiens | |||
| 19. | ALA4097298 | 25 | INH | = | 17 | % | ALA4016920 | % | Homo sapiens | |||
| 20. | ALA4097298 | 25 | INH | = | 8 | % | ALA4016921 | % | Homo sapiens |
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