| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4098390 | 5 | Time | = | 33 | min | ALA5233312 | hr | Mus musculus | |||
| 2. | ALA4098390 | 5 | Activity | = | 10.24 | mmHg | ALA5233311 | mmHg | Mus musculus | |||
| 3. | ALA4098390 | 5 | pEC50 | = | 8.37 | ALA5233310 | 8.37 | nM | Homo sapiens | |||
| 4. | ALA4098390 | 5 | pKi | = | 9.72 | ALA5233309 | 9.72 | nM | Rattus norvegicus | |||
| 5. | ALA4098390 | 5 | PPB | = | 57 | % | ALA5233308 | % | ||||
| 6. | ALA4098390 | 5 | t1/2 | = | 0.9 | hr | ALA5233306 | hr | ||||
| 7. | ALA4098390 | 5 | t1/2 | = | 10.95 | hr | ALA5233304 | hr | Homo sapiens | |||
| 8. | ALA4098390 | 5 | Activity | 0 | ALA4040240 | Toxic | Mus musculus | |||||
| 9. | ALA4098390 | 5 | Activity | 0 | ALA4040235 | Active | Mus musculus | |||||
| 10. | ALA4098390 | 5 | Ki | = | 0.19 | nM | ALA4040233 | 9.72 | nM | Rattus norvegicus | ||
| 11. | ALA4098390 | 5 | Drug degradation | = | 35 | % | ALA4040231 | % | Homo sapiens | |||
| 12. | ALA4098390 | 5 | Drug degradation | = | 43 | % | ALA4040230 | % | Homo sapiens | |||
| 13. | ALA4098390 | 5 | Drug metabolism | 0 | ALA4040229 | Metabolite_Detected | Homo sapiens | |||||
| 14. | ALA4098390 | 5 | EC50 | = | 4.1 | nM | ALA4401048 | 8.39 | nM | Homo sapiens | ||
| 15. | ALA4098390 | 5 | Activity | = | -32 | mmHg | ALA4401049 | mmHg | Mus musculus | |||
| 16. | ALA4098390 | 5 | Activity | 0 | ALA4401049 | Tde | Mus musculus | |||||
| 17. | ALA4098390 | 5 | Activity | 0 | ALA4401027 | Active | Homo sapiens | |||||
| 18. | ALA4098390 | 5 | Activity | 0 | ALA4401028 | Active | Homo sapiens | |||||
| 19. | ALA4098390 | 5 | Time | < | 1 | hr | ALA4401029 | hr | Homo sapiens | |||
| 20. | ALA4098390 | 5 | Time | < | 30 | min | ALA4401030 | hr | Homo sapiens |
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