# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4098390 | 5 | Time | = | 33 | min | ALA5233312 | hr | Mus musculus | |||
2. | ALA4098390 | 5 | Activity | = | 10.24 | mmHg | ALA5233311 | mmHg | Mus musculus | |||
3. | ALA4098390 | 5 | pEC50 | = | 8.37 | ALA5233310 | 8.37 | nM | Homo sapiens | |||
4. | ALA4098390 | 5 | pKi | = | 9.72 | ALA5233309 | 9.72 | nM | Rattus norvegicus | |||
5. | ALA4098390 | 5 | PPB | = | 57 | % | ALA5233308 | % | ||||
6. | ALA4098390 | 5 | t1/2 | = | 0.9 | hr | ALA5233306 | hr | ||||
7. | ALA4098390 | 5 | t1/2 | = | 10.95 | hr | ALA5233304 | hr | Homo sapiens | |||
8. | ALA4098390 | 5 | EC50 | = | 4.1 | nM | ALA4401048 | 8.39 | nM | Homo sapiens | ||
9. | ALA4098390 | 5 | Activity | = | -32 | mmHg | ALA4401049 | mmHg | Mus musculus | |||
10. | ALA4098390 | 5 | Activity | 0 | ALA4401049 | Tde | Mus musculus | |||||
11. | ALA4098390 | 5 | Activity | 0 | ALA4401027 | Active | Homo sapiens | |||||
12. | ALA4098390 | 5 | Activity | 0 | ALA4401028 | Active | Homo sapiens | |||||
13. | ALA4098390 | 5 | Time | < | 1 | hr | ALA4401029 | hr | Homo sapiens | |||
14. | ALA4098390 | 5 | Time | < | 30 | min | ALA4401030 | hr | Homo sapiens | |||
15. | ALA4098390 | 5 | Km | = | 30 | uM | ALA4401034 | nM | Homo sapiens | |||
16. | ALA4098390 | 5 | Kcat | = | 1.4 | /s | ALA4401035 | /s | Homo sapiens | |||
17. | ALA4098390 | 5 | Kcat/Km | = | 4.7 | 10'4/Ms | ALA4401036 | 10'4/Ms | Homo sapiens | |||
18. | ALA4098390 | 5 | Vmax | = | 0.316 | micromol/min | ALA4401043 | micromol/min | Homo sapiens | |||
19. | ALA4098390 | 5 | t1/2 | = | 1 | hr | ALA4401044 | hr | Homo sapiens | |||
20. | ALA4098390 | 5 | t1/2 | = | 0.7 | hr | ALA4401045 | hr | Homo sapiens |