# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4098822 | 1 | IC50 | = | 75 | nM | ALA4427245 | 7.12 | nM | Homo sapiens | ||
2. | ALA4098822 | 1 | solubility | = | 7 | ug ml-1 | ALA4427246 | ug.mL-1 | ||||
3. | ALA4098822 | 1 | solubility | = | 79 | ug ml-1 | ALA4427247 | ug.mL-1 | ||||
4. | ALA4098822 | 1 | Stability | > | 97 | % | ALA4427248 | % | ||||
5. | ALA4098822 | 1 | Stability | > | 97 | % | ALA4427249 | % | ||||
6. | ALA4098822 | 1 | IC50 | > | 40 | uM | ALA4427250 | nM | Homo sapiens | |||
7. | ALA4098822 | 1 | IC50 | > | 40 | uM | ALA4427251 | nM | Homo sapiens | |||
8. | ALA4098822 | 1 | IC50 | > | 40 | uM | ALA4427252 | nM | Homo sapiens | |||
9. | ALA4098822 | 1 | IC50 | > | 40 | uM | ALA4427253 | nM | Homo sapiens | |||
10. | ALA4098822 | 1 | IC50 | > | 40 | uM | ALA4427254 | nM | Homo sapiens | |||
11. | ALA4098822 | 1 | IC50 | > | 40 | uM | ALA4427255 | nM | Homo sapiens | |||
12. | ALA4098822 | 1 | IC50 | > | 40 | uM | ALA4427256 | nM | Homo sapiens | |||
13. | ALA4098822 | 1 | permeability | = | 37 | 10'-6 cm/s | ALA4427257 | 10'-6 cm/s | ||||
14. | ALA4098822 | 1 | Ratio | = | 1.2 | ALA4427258 | Homo sapiens | |||||
15. | ALA4098822 | 1 | Activity | 0 | ALA4427259 | Not Active | Homo sapiens | |||||
16. | ALA4098822 | 1 | Activity | 0 | ALA4427260 | Not Active | Homo sapiens | |||||
17. | ALA4098822 | 1 | IC50 | = | 15 | uM | ALA4427261 | 4.82 | nM | Homo sapiens | ||
18. | ALA4098822 | 1 | t1/2 | = | 9.2 | hr | ALA4427262 | hr | ||||
19. | ALA4098822 | 1 | CL | = | 2.3 | ml/min.kg | ALA4427263 | mL.min-1.kg-1 | ||||
20. | ALA4098822 | 1 | Vdss | = | 1.5 | L/Kg | ALA4427264 | L.kg-1 |