| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4101809 | 47 | Activity | = | 58 | % | ALA4839810 | % | Rattus norvegicus | |||
| 2. | ALA4101809 | 47 | Activity | = | 30 | % | ALA4839809 | % | Rattus norvegicus | |||
| 3. | ALA4101809 | 47 | Ratio | = | 0.7 | ALA4839808 | ||||||
| 4. | ALA4101809 | 47 | Activity | = | 43 | % | ALA4839807 | % | Mus musculus | |||
| 5. | ALA4101809 | 47 | Ratio | = | 1.1 | ALA4839806 | ||||||
| 6. | ALA4101809 | 47 | CL free | = | 51 | ml/min.kg | ALA4839805 | mL.min-1.kg-1 | ||||
| 7. | ALA4101809 | 47 | EC90 | = | 383 | nM | ALA4839804 | nM | Homo sapiens | |||
| 8. | ALA4101809 | 47 | EC50 | = | 35 | nM | ALA4839804 | 7.46 | nM | Homo sapiens | ||
| 9. | ALA4101809 | 47 | IC50 | = | 17 | uM | ALA4009621 | 4.77 | nM | Homo sapiens | ||
| 10. | ALA4101809 | 47 | IC50 | > | 25 | uM | ALA4009622 | nM | Homo sapiens | |||
| 11. | ALA4101809 | 47 | IC50 | = | 8 | uM | ALA4009623 | 5.10 | nM | Homo sapiens | ||
| 12. | ALA4101809 | 47 | IC50 | = | 2 | uM | ALA4009624 | 5.70 | nM | Homo sapiens | ||
| 13. | ALA4101809 | 47 | IC50 | = | 3 | uM | ALA4009625 | 5.52 | nM | Homo sapiens | ||
| 14. | ALA4101809 | 47 | Activity | 0 | ALA4009626 | Non-Toxic | Homo sapiens | |||||
| 15. | ALA4101809 | 47 | Activity | 0 | ALA4009627 | Non-Toxic | Homo sapiens | |||||
| 16. | ALA4101809 | 47 | AUClast | = | 67.8 | uM.hr | ALA4009610 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 17. | ALA4101809 | 47 | AUClast | = | 8.1 | uM.hr | ALA4009611 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Macaca fascicularis | ||
| 18. | ALA4101809 | 47 | Cmax | = | 7.3 | uM | ALA4009612 | nM | Rattus norvegicus | |||
| 19. | ALA4101809 | 47 | Cmax | = | 11 | uM | ALA4009613 | nM | Macaca fascicularis | |||
| 20. | ALA4101809 | 47 | F | = | 93 | % | ALA4009614 | % | Rattus norvegicus |
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