# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4102019 | 6 | INH | 0 | ALA4222566 | Active | % | Homo sapiens | ||||
2. | ALA4102019 | 6 | INH | 0 | ALA4222564 | Not Active | % | Homo sapiens | ||||
3. | ALA4102019 | 6 | INH | 0 | ALA4222563 | Not Active | % | Homo sapiens | ||||
4. | ALA4102019 | 6 | INH | 0 | ALA4222562 | Active | % | Homo sapiens | ||||
5. | ALA4102019 | 6 | INH | 0 | ALA4222561 | Not Active | % | Homo sapiens | ||||
6. | ALA4102019 | 6 | INH | 0 | ALA4222560 | Not Active | % | |||||
7. | ALA4102019 | 6 | INH | 0 | ALA4222559 | Not Active | % | Homo sapiens | ||||
8. | ALA4102019 | 6 | INH | 0 | ALA4222558 | Not Active | % | Homo sapiens | ||||
9. | ALA4102019 | 6 | INH | 0 | ALA4222557 | Active | % | Homo sapiens | ||||
10. | ALA4102019 | 6 | Activity | 0 | ALA4222556 | Active | Homo sapiens | |||||
11. | ALA4102019 | 6 | EC50 | > | 40 | uM | ALA4222555 | nM | Homo sapiens | |||
12. | ALA4102019 | 6 | EC50 | > | 40 | uM | ALA4222554 | nM | Homo sapiens | |||
13. | ALA4102019 | 6 | EC50 | = | 0.14 | uM | ALA4222553 | 6.85 | nM | Homo sapiens | ||
14. | ALA4102019 | 6 | Kd | = | 0.7 | uM | ALA4222547 | 6.16 | nM | Homo sapiens | ||
15. | ALA4102019 | 6 | permeability | > | 2200 | 10'-6 cm/s | ALA4222546 | 10'-6 cm/s | ||||
16. | ALA4102019 | 6 | solubility | = | 70 | uM | ALA4222545 | nM | ||||
17. | ALA4102019 | 6 | IC50 | = | 0.26 | uM | ALA4222544 | 6.58 | nM | Homo sapiens | ||
18. | ALA4102019 | 6 | CLH | = | 361 | ml/min.kg | ALA4024542 | mL.min-1.kg-1 | Mus musculus | |||
19. | ALA4102019 | 6 | t1/2 | = | 0.15 | hr | ALA4024541 | hr | Mus musculus |