# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4102551 | (1R,5R,9S)-15.HCl | EC50 | = | 761 | nM | ALA4038732 | 6.12 | nM | Homo sapiens | ||
2. | ALA4102551 | (1R,5R,9S)-15.HCl | EC50 | = | 901 | nM | ALA4038731 | 6.04 | nM | Rattus norvegicus | ||
3. | ALA4102551 | (1R,5R,9S)-15.HCl | INH | > | 50 | % | ALA4038730 | % | Rattus norvegicus | |||
4. | ALA4102551 | (1R,5R,9S)-15.HCl | INH | > | 50 | % | ALA4038729 | % | Rattus norvegicus | |||
5. | ALA4102551 | (1R,5R,9S)-15.HCl | INH | > | 50 | % | ALA4038728 | % | Rattus norvegicus | |||
6. | ALA4102551 | (1R,5R,9S)-15.HCl | Ratio EC50 | = | 40 | ALA4038725 | ||||||
7. | ALA4102551 | (1R,5R,9S)-15.HCl | Ratio EC50 | = | 47 | ALA4038724 | ||||||
8. | ALA4102551 | (1R,5R,9S)-15.HCl | EC50 | = | 19 | nM | ALA4038722 | 7.72 | nM | Rattus norvegicus | ||
9. | ALA4102551 | (1R,5R,9S)-15.HCl | Activity | = | 18 | % | ALA4038721 | % | Homo sapiens | |||
10. | ALA4102551 | (1R,5R,9S)-15.HCl | Ki | = | 1.99 | nM | ALA4038719 | 8.70 | nM | Rattus norvegicus | ||
11. | ALA4102551 | (1R,5R,9S)-15.HCl | Ki | = | 161 | nM | ALA4038716 | 6.79 | nM | Rattus norvegicus | ||
12. | ALA4102551 | (1R,5R,9S)-15.HCl | Ki | = | 29.9 | nM | ALA4038717 | 7.52 | nM | Rattus norvegicus | ||
13. | ALA4102551 | (1R,5R,9S)-15.HCl | Activity | = | 83 | % | ALA4038720 | % | Rattus norvegicus | |||
14. | ALA4102551 | (1R,5R,9S)-15.HCl | Activity | = | 50 | % | ALA4038718 | % | Rattus norvegicus |