# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4102566 | 31 | Ratio IC50/EC50 | > | 800 | ALA4004731 | ||||||
2. | ALA4102566 | 31 | IC50 | = | 4 | uM | ALA4004722 | 5.40 | nM | Homo sapiens | ||
3. | ALA4102566 | 31 | IC50 | = | 9200 | nM | ALA4004705 | 5.04 | nM | Homo sapiens | ||
4. | ALA4102566 | 31 | EC50 | = | 11 | nM | ALA4004692 | 7.96 | nM | Rattus norvegicus | ||
5. | ALA4102566 | 31 | %max | = | 13 | % | ALA4004695 | % | Rattus norvegicus | |||
6. | ALA4102566 | 31 | %max | = | 49 | % | ALA4004696 | % | Rattus norvegicus | |||
7. | ALA4102566 | 31 | EC50 | = | 0.49 | nM | ALA4004697 | 9.31 | nM | Rattus norvegicus | ||
8. | ALA4102566 | 31 | IC50 | = | 4 | uM | ALA3997250 | 5.40 | nM | Homo sapiens | ||
9. | ALA4102566 | 31 | Drug uptake | = | 81 | nM | ALA3997249 | nM | Mus musculus | |||
10. | ALA4102566 | 31 | Cp | = | 273 | nM | ALA3997248 | nM | Mus musculus | |||
11. | ALA4102566 | 31 | MED | = | 0.3 | mg kg-1 | ALA3997247 | mg kg-1 | Mus musculus | |||
12. | ALA4102566 | 31 | Emax | = | 49 | % | ALA3997246 | % | Rattus norvegicus | |||
13. | ALA4102566 | 31 | Emax | = | 13 | % | ALA3997245 | % | Rattus norvegicus | |||
14. | ALA4102566 | 31 | EC50 | > | 100 | uM | ALA3997244 | nM | Homo sapiens | |||
15. | ALA4102566 | 31 | EC50 | > | 100 | uM | ALA3997243 | nM | Homo sapiens | |||
16. | ALA4102566 | 31 | EC50 | > | 100 | uM | ALA3997242 | nM | Homo sapiens | |||
17. | ALA4102566 | 31 | Ratio IC50/EC50 | = | 840 | ALA3997241 | ||||||
18. | ALA4102566 | 31 | EC50 | = | 11 | nM | ALA3997239 | 7.96 | nM | Rattus norvegicus | ||
19. | ALA4102566 | 31 | IC50 | = | 9200 | nM | ALA3997240 | 5.04 | nM | Homo sapiens |