| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4103117 | 18; MM-589 | Ki | < | 1 | nM | ALA4017368 | nM | ||||
| 2. | ALA4103117 | 18; MM-589 | INH | 0 | ALA4017389 | Not Active | % | Homo sapiens | ||||
| 3. | ALA4103117 | 18; MM-589 | INH | 0 | ALA4017388 | Not Active | % | Homo sapiens | ||||
| 4. | ALA4103117 | 18; MM-589 | INH | 0 | ALA4017387 | Not Active | % | Homo sapiens | ||||
| 5. | ALA4103117 | 18; MM-589 | INH | 0 | ALA4017386 | Not Active | % | Homo sapiens | ||||
| 6. | ALA4103117 | 18; MM-589 | INH | 0 | ALA4017385 | Not Active | % | Homo sapiens | ||||
| 7. | ALA4103117 | 18; MM-589 | Stability | 0 | ALA4017384 | Stable | % | |||||
| 8. | ALA4103117 | 18; MM-589 | t1/2 | > | 60 | min | ALA4017383 | hr | ||||
| 9. | ALA4103117 | 18; MM-589 | t1/2 | > | 60 | min | ALA4017382 | hr | ||||
| 10. | ALA4103117 | 18; MM-589 | t1/2 | > | 60 | min | ALA4017381 | hr | ||||
| 11. | ALA4103117 | 18; MM-589 | GI | > | 95 | % | ALA4017380 | % | Homo sapiens | |||
| 12. | ALA4103117 | 18; MM-589 | GI | > | 95 | % | ALA4017379 | % | Homo sapiens | |||
| 13. | ALA4103117 | 18; MM-589 | GI | = | 75 | % | ALA4017378 | % | Homo sapiens | |||
| 14. | ALA4103117 | 18; MM-589 | GI | = | 75 | % | ALA4017377 | % | Homo sapiens | |||
| 15. | ALA4103117 | 18; MM-589 | IC50 | = | 0.1 | uM | ALA4017376 | 7.00 | nM | Homo sapiens | ||
| 16. | ALA4103117 | 18; MM-589 | IC50 | = | 0.29 | uM | ALA4017375 | 6.54 | nM | Homo sapiens | ||
| 17. | ALA4103117 | 18; MM-589 | Ratio IC50 | > | 30 | ALA4017374 | ||||||
| 18. | ALA4103117 | 18; MM-589 | Ratio IC50 | > | 30 | ALA4017373 | ||||||
| 19. | ALA4103117 | 18; MM-589 | IC50 | = | 8.56 | uM | ALA4017372 | 5.07 | nM | Homo sapiens | ||
| 20. | ALA4103117 | 18; MM-589 | IC50 | = | 0.25 | uM | ALA4017371 | 6.60 | nM | Homo sapiens |
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