# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4104658 | 8 | AUClast | = | 466 | hr.ng/ml | ALA5238853 | ng.hr.mL-1 | ||||
2. | ALA4104658 | 8 | Cmax | = | 126 | ng/ml | ALA5238852 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
3. | ALA4104658 | 8 | AUClast | = | 285 | hr.ng/ml | ALA5238851 | ng.hr.mL-1 | ||||
4. | ALA4104658 | 8 | Cmax | = | 81 | ng/ml | ALA5238850 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
5. | ALA4104658 | 8 | IC50 | = | 405 | nM | ALA5238849 | 6.39 | nM | Homo sapiens | ||
6. | ALA4104658 | 8 | IC50 | = | 197 | nM | ALA5238848 | 6.71 | nM | |||
7. | ALA4104658 | 8 | IC50 | = | 54 | nM | ALA5238847 | 7.27 | nM | |||
8. | ALA4104658 | 8 | INH | = | 90 | % | ALA4053919 | % | Homo sapiens | |||
9. | ALA4104658 | 8 | INH | = | 14 | % | ALA4053918 | % | Homo sapiens | |||
10. | ALA4104658 | 8 | INH | = | 75 | % | ALA4053917 | % | Homo sapiens | |||
11. | ALA4104658 | 8 | INH | = | 52 | % | ALA4053916 | % | Homo sapiens | |||
12. | ALA4104658 | 8 | INH | = | 117 | % | ALA4053915 | % | Homo sapiens | |||
13. | ALA4104658 | 8 | INH | = | 110 | % | ALA4053914 | % | ||||
14. | ALA4104658 | 8 | INH | = | 10 | % | ALA4053913 | % | Homo sapiens | |||
15. | ALA4104658 | 8 | INH | = | 14 | % | ALA4053912 | % | Homo sapiens | |||
16. | ALA4104658 | 8 | INH | = | 88 | % | ALA4053911 | % | Homo sapiens | |||
17. | ALA4104658 | 8 | INH | = | 4 | % | ALA4053910 | % | Homo sapiens | |||
18. | ALA4104658 | 8 | INH | = | 72 | % | ALA4053909 | % | Homo sapiens | |||
19. | ALA4104658 | 8 | INH | = | 16 | % | ALA4053908 | % | Homo sapiens | |||
20. | ALA4104658 | 8 | INH | = | 10 | % | ALA4053907 | % | Homo sapiens |